SCHEMBL8199368

SCHEMBL8199368

O=C1c2ccc(OCc3ccccc3-c3ccccc3)cc2CCC1CCN1CCC(c2ccccc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 2/20 0.49
ADRA1D P25100 1/20 0.47
ADRA1A P35348 1/20 0.47
ADRA1B P35368 1/20 0.47
HTR7 P34969 2/20 0.46
CYP24A1 Q07973 5/20 0.44
CYP27A1 Q02318 3/20 0.44
HTR2C P28335 3/20 0.43
DRD2 P14416 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2B P41595 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
BACE1 P56817 1/20 0.41
CD274 Q9NZQ7 3/20 0.41
MAOB P27338 2/20 0.41
MAOA P21397 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8200598 0.90 CYP26A1 (0.52) CYP26A1HTR7CYP24A1CYP27A1HTR2C
SCHEMBL8205161 0.90 CYP24A1 (0.55) CYP26A1ADRA1DADRA1AADRA1BHTR7
SCHEMBL8204770 0.90 ADRA1D (0.47) CYP26A1ADRA1DADRA1AADRA1BHTR7
SCHEMBL8200537 0.89 ADRA1D (0.56) CYP26A1ADRA1DADRA1AADRA1BHTR7
SCHEMBL8198852 0.88 ADRA1D (0.57) CYP26A1ADRA1DADRA1AADRA1BHTR7
SCHEMBL8201758 0.88 HTR2C (0.52) CYP26A1ADRA1DADRA1AADRA1BHTR7
SCHEMBL8200296 0.87 ADRA1D (0.50) CYP26A1ADRA1DADRA1AADRA1BHTR7
SCHEMBL8198844 0.86 GPR84 (0.47) CYP26A1ADRA1DADRA1AADRA1BHTR7
SCHEMBL8200489 0.85 CYP24A1 (0.48) CYP26A1ADRA1DADRA1AADRA1BHTR7
SCHEMBL8204752 0.84 HTR7 (0.47) CYP26A1ADRA1DADRA1AADRA1BHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US claimed
WO-1998036749-A1 TETRALONE DERIVATIVES AS ANTIARRHYTHMIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-08-27 WO claimed
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed
WO-1998036749-A1 TETRALONE DERIVATIVES AS ANTIARRHYTHMIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-08-27 WO disclosed