SCHEMBL8201250

SCHEMBL8201250

N#CNC(=N)N(Cc1ccc(C(N)=O)cc1)c1ccncc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.43
MAPK14 Q16539 1/20 0.40
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
KMT2A Q03164 1/20 0.36
NAMPT P43490 3/20 0.35
IKBKE Q14164 1/20 0.35
TBK1 Q9UHD2 1/20 0.35
GAA P10253 1/20 0.33
TSHR P16473 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
PDK1 Q15118 1/20 0.33
KDM1A O60341 1/20 0.33
ABHD6 Q9BV23 1/20 0.33
CHUK O15111 1/20 0.33
INSR P06213 1/20 0.33
MAPK8 P45983 1/20 0.33
CAMKK2 Q96RR4 1/20 0.33
LTB4R2 Q9NPC1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7978140 0.74 CYP17A1 (0.43) CYP17A1MEN1NPC1KMT2ANAMPT
SCHEMBL8195511 0.73 HTT (0.55) MEN1KMT2ANAMPTPOLB
SCHEMBL8200235 0.67 CYP17A1 (0.46) CYP17A1NAMPT
SCHEMBL7902116 0.67 SIGMAR1 (0.40) NAMPTHDAC1
SCHEMBL1336855 0.66 TSHR (0.49) MAPK14MEN1NPC1KMT2AGAA
SCHEMBL23905177 0.65 CYP17A1 (0.89) CYP17A1MEN1KMT2ATSHRHDAC1
SCHEMBL27536266 0.65 CYP17A1 (0.71) CYP17A1NPC1HDAC1
Water SCHEMBL31094001 0.64 CYP17A1 (0.57) CYP17A1MEN1KMT2AGAATSHR
SCHEMBL27644588 0.64 MAPK14 (0.43) MAPK14NAMPTPDK1
SCHEMBL14716527 0.62 CYP17A1 (0.49) CYP17A1KMT2AGAATSHRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000061561-A1 CYANOGUANIDINE COMPOUNDS SHIONOGI BIORESEARCH CORP. (US) 2000-10-19 WO claimed