SCHEMBL8201273

SCHEMBL8201273

O=C(O)c1ccc(NC(=O)c2ccc3c(c2)CCC(CCN2CCC(c4ccccc4)CC2)C3=O)cc1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 5/20 0.48
ITGB3 P05106 2/20 0.46
ITGA2B P08514 2/20 0.46
MCHR1 Q99705 3/20 0.45
ACHE P22303 2/20 0.44
DGAT1 O75907 1/20 0.44
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
SIGMAR1 Q99720 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8204772 0.95 HTR2C (0.50) HTR2CITGB3ITGA2BMCHR1ACHE
SCHEMBL8192524 0.91 HTR2C (0.47) HTR2CITGB3ITGA2BMCHR1ACHE
SCHEMBL8198980 0.90 HTR2C (0.55) HTR2CMCHR1SIGMAR1
SCHEMBL8199033 0.89 HTR2C (0.46) HTR2CITGB3ITGA2BMCHR1ACHE
SCHEMBL8198493 0.88 MAPT (0.47) HTR2CITGB3ITGA2BMCHR1ACHE
SCHEMBL8198779 0.88 HTR2C (0.47) HTR2CITGB3ITGA2BACHE
SCHEMBL8200256 0.88 NAMPT (0.47) HTR2CITGB3ITGA2BACHELMNA
SCHEMBL8200675 0.86 HTR2C (0.49) HTR2CMCHR1
SCHEMBL8204780 0.86 ACHE (0.44) HTR2CITGB3ITGA2BMCHR1ACHE
SCHEMBL8204778 0.86 ACHE (0.44) HTR2CITGB3ITGA2BMCHR1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US claimed
WO-1998036749-A1 TETRALONE DERIVATIVES AS ANTIARRHYTHMIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-08-27 WO claimed
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed