SCHEMBL8201535

SCHEMBL8201535

Bc1cnc(C#N)nc1N(NC(=O)c1ccc(CN2CCN(CC3CCN(C)CC3)CC2)cc1)C1CCCCC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 7/20 0.55
CTSK P43235 6/20 0.55
CTSL P07711 5/20 0.55
CTSB P07858 1/20 0.55
PRKAA2 P54646 3/20 0.39
TBK1 Q9UHD2 2/20 0.38
HDAC6 Q9UBN7 1/20 0.38
IKBKE Q14164 1/20 0.35
HIF1A Q16665 1/20 0.35
EPAS1 Q99814 1/20 0.35
KIT P10721 1/20 0.35
FLT3 P36888 1/20 0.35
PRKAB2 O43741 1/20 0.35
PRKAG1 P54619 1/20 0.35
PRKAA1 Q13131 1/20 0.35
PRKAG3 Q9UGI9 1/20 0.35
PRKAG2 Q9UGJ0 1/20 0.35
PRKAB1 Q9Y478 1/20 0.35
ABL1 P00519 2/20 0.35
KLKB1 P03952 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8201088 0.94 CTSS (0.59) CTSSCTSKCTSLCTSBPRKAA2
SCHEMBL14142807 0.94 CTSS (0.53) CTSSCTSKCTSLCTSBPRKAA2
SCHEMBL14142811 0.93 CTSS (0.60) CTSSCTSKCTSLCTSBPRKAA2
SCHEMBL14142826 0.91 CTSS (0.46) CTSSCTSKCTSLCTSBKLKB1
SCHEMBL8205409 0.91 CTSS (0.52) CTSSCTSKCTSLCTSBPRKAA2
SCHEMBL3180410 0.91 CTSS (0.65) CTSSCTSKCTSLCTSBPRKAA2
SCHEMBL3165989 0.90 CTSS (0.66) CTSSCTSKCTSLCTSBPRKAA2
SCHEMBL14142757 0.90 CTSS (0.54) CTSSCTSKCTSLCTSBPRKAA2
SCHEMBL8245361 0.89 CTSS (0.58) CTSSCTSKCTSLCTSBPRKAA2
SCHEMBL14142743 0.88 CTSS (0.53) CTSSCTSKCTSLCTSBPRKAA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008052934-A1 NOVEL SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2008-05-08 WO disclosed