SCHEMBL8205409

SCHEMBL8205409

Bc1cnc(C#N)nc1N(NC(=O)c1ccc(CN2CCN(CC3CCN(C)CC3)CC2)cc1)C1CCC(C)C1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 4/20 0.52
CTSK P43235 4/20 0.52
CTSL P07711 3/20 0.52
CTSB P07858 1/20 0.52
TBK1 Q9UHD2 2/20 0.36
HDAC6 Q9UBN7 1/20 0.35
CHRM4 P08173 3/20 0.34
IKBKE Q14164 1/20 0.34
CHRM2 P08172 2/20 0.34
CHRM1 P11229 2/20 0.34
PRKAA2 P54646 3/20 0.33
ABL1 P00519 3/20 0.33
PRKAB2 O43741 1/20 0.33
PRKAG1 P54619 1/20 0.33
PRKAA1 Q13131 1/20 0.33
PRKAG3 Q9UGI9 1/20 0.33
PRKAG2 Q9UGJ0 1/20 0.33
PRKAB1 Q9Y478 1/20 0.33
KIT P10721 1/20 0.33
FLT3 P36888 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14142812 0.92 CTSS (0.53) CTSSCTSKCTSLCTSBTBK1
SCHEMBL3169601 0.92 CTSS (0.62) CTSSCTSKCTSLCTSBTBK1
SCHEMBL8201535 0.91 CTSS (0.55) CTSSCTSKCTSLCTSBTBK1
SCHEMBL14142807 0.89 CTSS (0.53) CTSSCTSKCTSLCTSBTBK1
SCHEMBL14142814 0.89 CTSS (0.51) CTSSCTSKCTSLCTSBTBK1
Trifluoroacetic Acid SCHEMBL3160152 0.87 CTSS (0.57) CTSSCTSKCTSLCTSBTBK1
SCHEMBL14142811 0.86 CTSS (0.60) CTSSCTSKCTSLCTSBTBK1
SCHEMBL3169883 0.85 CTSS (0.67) CTSSCTSKCTSLCTSBTBK1
SCHEMBL8201088 0.85 CTSS (0.59) CTSSCTSKCTSLCTSBTBK1
SCHEMBL8245361 0.83 CTSS (0.58) CTSSCTSKCTSLCTSBTBK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008052934-A1 NOVEL SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2008-05-08 WO disclosed