SCHEMBL8201592

SCHEMBL8201592

COc1ccc(C(=O)n2cc(C[C@H]3CCCN3C)c3cc(Cl)ccc32)cc1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 14/20 0.56
AKR1C2 P52895 9/20 0.56
PTGS1 P23219 2/20 0.56
AKR1C4 P17516 1/20 0.56
HTR6 P50406 2/20 0.53
AR P10275 1/20 0.48
PTGS2 P35354 2/20 0.46
HTR1A P08908 1/20 0.46
HTR1B P28222 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8201597 1.00 AKR1C3 (0.56) AKR1C3AKR1C2PTGS1AKR1C4HTR6
SCHEMBL8208572 0.89 HTR6 (0.55) AKR1C3AKR1C2PTGS1AKR1C4HTR6
SCHEMBL8208569 0.89 HTR6 (0.55) AKR1C3AKR1C2PTGS1AKR1C4HTR6
SCHEMBL8209785 0.89 HTR6 (0.64) AKR1C3AKR1C2PTGS1AKR1C4HTR6
SCHEMBL8209782 0.89 HTR6 (0.64) AKR1C3AKR1C2PTGS1AKR1C4HTR6
SCHEMBL8208554 0.87 HTR6 (0.64) HTR6
SCHEMBL8213128 0.87 HTR6 (0.64) HTR6
SCHEMBL8209078 0.86 HTR6 (0.55) AKR1C3AKR1C2PTGS1AKR1C4HTR6
SCHEMBL8209082 0.86 HTR6 (0.55) AKR1C3AKR1C2PTGS1AKR1C4HTR6
SCHEMBL8201580 0.80 HTR6 (0.79) HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6100291-A FOR TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS ALLELIX BIOPHARMACEUTICALS INC. (CA) 2000-08-08 US disclosed
WO-1999047516-A1 3-(2-PYRROLIDINYLMETHYL)-INDOLE COMPOUNDS HAVING 5-HT6 AFFINITY SLASSI ABDELMALIK (CA) 1999-09-23 WO disclosed