SCHEMBL8201619

SCHEMBL8201619

c1ccc(CCCc2ccc(P(Cc3ccccc3-c3ccccc3CP(c3ccc(CCCc4ccccc4)cc3)c3ccc(CCCc4ccccc4)cc3)c3ccc(CCCc4ccccc4)cc3)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.44
MAOB P27338 2/20 0.40
SIGMAR1 Q99720 3/20 0.37
MAOA P21397 1/20 0.37
HDAC8 Q9BY41 2/20 0.37
HDAC1 Q13547 2/20 0.37
IGF1R P08069 1/20 0.36
ALOX15 P16050 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PTGER1 P34995 1/20 0.35
PTGER4 P35408 1/20 0.35
PTGER3 P43115 1/20 0.35
PTGER2 P43116 1/20 0.35
IDO1 P14902 1/20 0.35
HDAC3 O15379 1/20 0.35
MAPK1 P28482 1/20 0.35
ADRA1A P35348 1/20 0.35
HDAC4 P56524 1/20 0.35
SLC6A3 Q01959 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8203447 0.82 SMN1; SMN2 (0.36) HDAC8HDAC1SMN1; SMN2
SCHEMBL720169 0.81 CYP3A4 (0.38) TDP1PTGER1PTGER4PTGER3PTGER2
SCHEMBL29695439 0.79 CYP3A4 (0.36) TDP1PTGER1PTGER4PTGER3PTGER2
Phosphine SCHEMBL29173742 0.79 CYP3A4 (0.36) TDP1PTGER1PTGER4PTGER3PTGER2
Lithium SCHEMBL29695298 0.79 CYP3A4 (0.36) TDP1PTGER1PTGER4PTGER3PTGER2
Potassium SCHEMBL30843013 0.79 CYP3A4 (0.36) TDP1PTGER1PTGER4PTGER3PTGER2
Bromide SCHEMBL30945893 0.77 CYP3A4 (0.35) TDP1
SCHEMBL19002937 0.76 CSNK2A2 (0.30)
SCHEMBL8056033 0.75 PTGS2 (0.33) TDP1
SCHEMBL30945894 0.74 DPP4 (0.32) TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043398-A WATER-SOLUBLE, SULFONATED DIPHOSPHINES COMPLEXED WITH A TRANSITION METAL TO FORM HYDROFORMYLATION CATALYSTS; OUTSTANDING SURFACE ACTIVE PROPERTIES IN TWO PHASE CATALYSIS OF TWO PHASE HYDROFORMYLATION OF OCT-1-ENE OLEFINS CELANESE INTERNATIONAL CORPORATION (US) 2000-03-28 US disclosed