SCHEMBL8201683

SCHEMBL8201683

C[S+]([O-])c1ccc(-c2[nH]nc(C(F)(F)F)c2-c2ccc(F)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 4/20 0.44
PTGS2 P35354 7/20 0.33
ENPP1 P22413 1/20 0.33
GYS1 P13807 1/20 0.33
MAPK1 P28482 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
MAPT P10636 2/20 0.32
MAPK13 O15264 1/20 0.31
MAPK12 P53778 1/20 0.31
MAPK11 Q15759 1/20 0.31
RPS6KA3 P51812 1/20 0.31
PTGS1 P23219 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8196073 0.90 ENPP1 (0.35) MAPK14PTGS2ENPP1MAPK1NPSR1
SCHEMBL8642544 0.83
SCHEMBL8637992 0.81 MAPK14 (0.46) MAPK14PTGS2MAPK1NPSR1MAPK13
SCHEMBL8201927 0.81 IKBKE (0.39) PTGS2MAPK1RPS6KA3
SCHEMBL5078441 0.80 PTGS2 (0.53) MAPK14PTGS2MAPK11PTGS1
SCHEMBL6180483 0.80 PTGS2 (0.53) MAPK14PTGS2MAPK11PTGS1
SCHEMBL14519434 0.79 MAPK14 (0.64) MAPK14MAPK13MAPK12MAPK11
SCHEMBL4212020 0.79 PTGS2 (0.52) MAPK14PTGS2MAPK11PTGS1
SCHEMBL8194882 0.78 PTGS2 (0.38) PTGS2PTGS1
SCHEMBL8194744 0.76 MAPK14 (0.41) MAPK14PTGS2ENPP1GYS1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO disclosed