SCHEMBL8202019

SCHEMBL8202019

NCC(=O)N1CCCC1CN[C@@H](Cc1ccccc1)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.49
HSD17B10 Q99714 1/20 0.49
ACE P12821 6/20 0.47
DPP4 P27487 6/20 0.46
DPP8 Q6V1X1 4/20 0.46
DPP7 Q9UHL4 4/20 0.46
DPP9 Q86TI2 3/20 0.46
FAP Q12884 1/20 0.46
ATM Q13315 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
ACE2 Q9BYF1 1/20 0.44
POLB P06746 1/20 0.43
ITGB1 P05556 1/20 0.43
ITGA4 P13612 1/20 0.43
ITGB7 P26010 1/20 0.43
F2 P00734 1/20 0.42
PRSS1 P07477 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8191997 0.85 DPP4 (0.61) DPP4DPP8DPP7DPP9FAP
SCHEMBL30050973 0.80 ITGB1 (0.57) ALDH1A1HSD17B10ACEACE2ITGB1
SCHEMBL29743032 0.75 SLC6A2 (0.52) ACEF2
SCHEMBL6302781 0.72 ITGB1 (0.59) ALDH1A1ITGB1ITGA4ITGB7
SCHEMBL9074016 0.72 ACE (0.50) ALDH1A1HSD17B10ACEATML3MBTL1
SCHEMBL9074014 0.72 ACE (0.50) ALDH1A1HSD17B10ACEATML3MBTL1
SCHEMBL30563223 0.71 ACE (0.53) ACEITGB1F2
SCHEMBL30862234 0.71 SLC6A2 (0.54) ACEITGB1
SCHEMBL10903563 0.71 ACE2 (0.56) L3MBTL1ACE2
SCHEMBL10903562 0.71 ACE2 (0.56) L3MBTL1ACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6090786-A HALOPYRROLE AMIDATED AMINO ACID USEFUL FOR INHIBITING SERINE PROTEASE ACTIVITY FONDATECH BENELUX N.V. (BE) 2000-07-18 US disclosed
EP-0764151-A2 PURIFICATION OF SERINE PROTEASE AND SYNTHETIC INHIBITORS THEREOF UNIVERSITAIRE INSTELLING ANTWERPEN (BE) 1997-03-26 EP disclosed
WO-1995034538-A2 PURIFICATION OF SERINE PROTEASES AND SYNTHETIC INHIBITORS THEREOF UNIVERSITAIRE INSTELLING ANTWERPEN (BE) 1995-12-21 WO disclosed