SCHEMBL8202497

SCHEMBL8202497

O=C1Nc2ccccc2Nc2ccc(C(F)(F)F)cc21

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACVR1 Q04771 2/20 0.58
LRRK2 Q5S007 2/20 0.58
CDK5 Q00535 2/20 0.58
ROS1 P08922 1/20 0.58
PDGFRA P16234 1/20 0.56
FER P16591 1/20 0.56
LTK P29376 1/20 0.56
CDK8 P49336 1/20 0.56
DYRK1B Q9Y463 1/20 0.56
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
GALR3 O60755 1/20 0.52
CSNK1G1 Q9HCP0 1/20 0.51
CHEK1 O14757 1/20 0.51
JUN P05412 3/20 0.49
NFKB1 P19838 3/20 0.49
NFKB2 Q00653 3/20 0.49
RELA Q04206 3/20 0.49
CYBB P04839 1/20 0.47
NOX3 Q9HBY0 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29486043 0.87 ACVR1 (0.56) ACVR1LRRK2CDK5ROS1PDGFRA
SCHEMBL22748875 0.87 ACVR1 (0.56) ACVR1LRRK2CDK5ROS1PDGFRA
SCHEMBL20442582 0.84 CSNK1G1 (0.61) ACVR1LRRK2CDK5ROS1PDGFRA
SCHEMBL2372316 0.81 CES1 (0.58) GALR3JUNNFKB1NFKB2RELA
SCHEMBL30120589 0.81 CES1 (0.58) GALR3JUNNFKB1NFKB2RELA
SCHEMBL14365137 0.80 CYBB (0.47) ACVR1LRRK2CDK5ROS1PDGFRA
Hydrochloric Acid SCHEMBL11435666 0.79 CES1 (0.57) GALR3JUNNFKB1NFKB2RELA
SCHEMBL3616249 0.77 LRRK2 (0.64) ACVR1LRRK2CDK5ROS1PDGFRA
SCHEMBL31098215 0.77 ACE2 (0.56) MEN1KMT2AGALR3JUNNFKB1
Toluene SCHEMBL28093752 0.77 MAOA (0.51) ACVR1LRRK2CDK5ROS1GALR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6103715-A COMPOUNDS THAT BIND TO THE DOPAMINE D4 RECEPTOR AND THEIR USE AS ANXIOLYTIC AGENTS, TREATMENT FOR SCHIZOPHRENIA, AND DRUG SCREENING; SIDE EFFECT REDUCTIOON ALLELIX BIOPHARMACEUTICALS INC. (CA) 2000-08-15 US disclosed
US-5968478-A DIBENZOTHIEPINE AS NEUROTRANSMITTERS AND FOR DRUG SCREENING AND TREATMENT OF SCHIZOPHRENIA ALLELIX BIOPHARMACEUTICALS, INC. (CA) 1999-10-19 US disclosed