SCHEMBL8203062

SCHEMBL8203062

C/C=C/c1cc2c(O[C@@H]3C[C@@H](C(=O)OC)N(C(=O)[C@@H](NC(=O)OC4CCCC4)C4CCCC4)C3)cc(OCC)nc2cc1OC

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSB P07858 1/20 0.35
PPP3CB P16298 1/20 0.35
ELANE P08246 1/20 0.33
KCNH2 Q12809 1/20 0.33
HTR3E A5X5Y0 1/20 0.32
HTR3B O95264 1/20 0.32
HTR3A P46098 1/20 0.32
HTR3D Q70Z44 1/20 0.32
HTR3C Q8WXA8 1/20 0.32
CYP3A4 P08684 1/20 0.31
EGFR P00533 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8203717 0.95 CTSB (0.36) CTSBPPP3CBELANEKCNH2HTR3E
SCHEMBL13402558 0.84 CTSB (0.33) CTSBPPP3CBELANEKCNH2EGFR
SCHEMBL3496929 0.80 CTSB (0.34) CTSBPPP3CBELANEKCNH2HTR3E
SCHEMBL1072404 0.79 PDE4B (0.33) CTSBPPP3CBCYP3A4EGFR
SCHEMBL13437245 0.76 CTSB (0.30) CTSBPPP3CB
SCHEMBL14092828 0.76 CTSB (0.55) CTSBPPP3CBCYP3A4
SCHEMBL15397439 0.75 PDE4B (0.33) CTSBPPP3CBCYP3A4
SCHEMBL20292518 0.75 PDE4B (0.33) CTSBPPP3CBCYP3A4
SCHEMBL2754150 0.74 AAK1 (0.38) CTSBPPP3CBELANEKCNH2CYP3A4
SCHEMBL12934499 0.73 P2RX3 (0.39) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008051514-A2 HCV NS3 PROTEASE INHIBITORS MERCK & CO., INC. (US) 2008-05-02 WO disclosed