SCHEMBL8203558

SCHEMBL8203558

CC(C)(C)CCNC(=O)c1ccc2c(c1)CCCC2=O

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 1/20 0.48
BAZ2B Q9UIF8 1/20 0.47
NAMPT P43490 3/20 0.46
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
PRKCI P41743 1/20 0.44
MAPK14 Q16539 7/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 1/20 0.42
HSD17B1 P14061 1/20 0.41
PARP10 Q53GL7 1/20 0.41
S1PR1 P21453 1/20 0.40
S1PR3 Q99500 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8589013 0.84 MLYCD (0.45) MLYCDNAMPTNPC1RAB9AKMT2A
SCHEMBL8589012 0.84 MLYCD (0.45) MLYCDNAMPTNPC1RAB9AKMT2A
SCHEMBL22500097 0.79 MAPK1 (0.56) BAZ2BMAOAMAOBPRKCIMAPK14
SCHEMBL22516823 0.79 MAPK14 (0.49) BAZ2BMAOAMAOBPRKCIMAPK14
SCHEMBL19029127 0.78 BAZ2B (0.56) BAZ2BMAOAMAOBPRKCIMAPK14
SCHEMBL29649324 0.78 BAZ2B (0.56) BAZ2BMAOAMAOBPRKCIMAPK14
SCHEMBL22500434 0.78 MAPK1 (0.58) BAZ2BMAOAMAOBPRKCIMAPK14
SCHEMBL22517131 0.78 MAPK14 (0.48) BAZ2BMAPK14NPC1RAB9A
SCHEMBL8201692 0.76 MLYCD (0.42) MLYCDNAMPTMAPK14KMT2AS1PR1
SCHEMBL8198550 0.76 MLYCD (0.46) MLYCDNAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998036749-A1 TETRALONE DERIVATIVES AS ANTIARRHYTHMIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-08-27 WO claimed
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed
WO-1998036749-A1 TETRALONE DERIVATIVES AS ANTIARRHYTHMIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-08-27 WO disclosed