SCHEMBL8201692

SCHEMBL8201692

CCCC1CCc2cc(C(=O)NCCC(C)(C)C)ccc2C1=O

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 1/20 0.42
NAMPT P43490 3/20 0.41
ITGB3 P05106 7/20 0.41
ITGA2B P08514 7/20 0.41
CYP26A1 O43174 1/20 0.37
MAPK14 Q16539 1/20 0.37
SGPL1 O95470 1/20 0.37
S1PR1 P21453 1/20 0.37
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8192821 0.92 THRA (0.42) MLYCDNAMPTITGB3ITGA2BMAPK14
SCHEMBL8198845 0.85 MLYCD (0.40) MLYCDNAMPTITGB3ITGA2BCYP26A1
SCHEMBL8200547 0.81 HTR2C (0.48) NAMPT
SCHEMBL8205603 0.78 SMN1; SMN2 (0.48) MAPK14MAPTKMT2A
SCHEMBL8203558 0.76 MLYCD (0.48) MLYCDNAMPTMAPK14S1PR1KMT2A
SCHEMBL8588802 0.73 HTR2C (0.48) TP53MAPTTHRB
SCHEMBL8199839 0.72 MLYCD (0.45) MLYCDNAMPTSGPL1S1PR1THRB
SCHEMBL8199972 0.72 HTR2C (0.46) KMT2A
SCHEMBL8589013 0.71 MLYCD (0.45) MLYCDNAMPTTP53MAPTKMT2A
SCHEMBL8589012 0.71 MLYCD (0.45) MLYCDNAMPTTP53MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998036749-A1 TETRALONE DERIVATIVES AS ANTIARRHYTHMIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-08-27 WO claimed
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed