SCHEMBL8204092

SCHEMBL8204092

Cc1nc2c(n1C)CCN(C(=O)c1ccc(NC(=O)c3ccccc3-c3ccccc3)cc1)c1ccccc1-2

nearest known ligand 0.74

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 16/20 0.74
AVPR1A P37288 11/20 0.74
AVPR1B P47901 4/20 0.60
OXTR P30559 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6993733 0.99 AVPR2 (0.73) AVPR2AVPR1AAVPR1BOXTR
SCHEMBL10109005 0.90 AVPR2 (0.70) AVPR2AVPR1AAVPR1BOXTR
SCHEMBL17471541 0.87 AVPR2 (0.68) AVPR2AVPR1AAVPR1BOXTR
Conivaptan SCHEMBL49815 0.85 AVPR2 (1.00) AVPR2AVPR1AAVPR1BOXTR
SCHEMBL6991859 0.85 AVPR1A (0.72) AVPR2AVPR1AAVPR1BOXTR
Conivaptan SCHEMBL28043077 0.84 AVPR2 (0.98) AVPR2AVPR1AAVPR1BOXTR
Conivaptan SCHEMBL1649913 0.83 AVPR2 (0.97) AVPR2AVPR1AAVPR1BOXTR
SCHEMBL6619403 0.81 AVPR2 (0.65) AVPR2AVPR1AAVPR1BOXTR
SCHEMBL6995135 0.80 AVPR2 (0.48) AVPR2AVPR1AOXTR
Conivaptan SCHEMBL4625101 0.80 AVPR2 (0.75) AVPR2AVPR1AAVPR1BOXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008097546-A2 COMPOUNDS THAT INHIBIT CHOLINESTERASE COLUCID PHARMACEUTICALS, INC. (US) 2008-08-14 WO disclosed