SCHEMBL8205035

SCHEMBL8205035

O=C1NC(=O)C2(CCNCC2)N1c1cccc(F)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.44
MGLL Q99685 1/20 0.44
HSD17B10 Q99714 1/20 0.43
ALDH1A1 P00352 3/20 0.41
BACE1 P56817 2/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
USP2 O75604 2/20 0.40
CYP2D6 P10635 2/20 0.40
ALOX5 P09917 2/20 0.40
ALOX15 P16050 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CYP2C19 P33261 1/20 0.39
MCHR1 Q99705 1/20 0.39
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8808180 0.82 HSD17B10 (0.41) MGLLHSD17B10ALDH1A1POLBMAPT
SCHEMBL8204221 0.82 ALOX5 (0.43) FAAHMGLLALDH1A1BACE1POLB
SCHEMBL8811652 0.82 HSD17B10 (0.58) HSD17B10ALDH1A1BACE1USP2CYP2D6
Hydrochloric Acid SCHEMBL8809755 0.81 HSD17B10 (0.40) MGLLHSD17B10ALDH1A1MAPTMCHR1
SCHEMBL592180 0.78 ALDH1A1 (0.37) FAAHMGLLHSD17B10ALDH1A1BACE1
SCHEMBL8209542 0.77 BACE1 (0.67) BACE1CYP2D6MCHR1OPRM1OPRD1
SCHEMBL30436420 0.77 BACE1 (0.43) FAAHMGLLALDH1A1BACE1POLB
SCHEMBL25258942 0.75 AR (0.55) FAAHMGLLALDH1A1POLBGAA
SCHEMBL30381901 0.75 AR (0.55) FAAHMGLLALDH1A1POLBGAA
Trifluoroacetic Acid SCHEMBL4252943 0.75 ALOX5 (0.38) ALDH1A1BACE1USP2CYP2D6ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008030412-A2 SPIROPIPERIDINE BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE MERCK & CO., INC. (US) 2008-03-13 WO disclosed