SCHEMBL8205073

SCHEMBL8205073

COC(=O)Cc1n[nH]c2cc(F)cc(F)c12

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.45
MAPT P10636 1/20 0.44
MAP2K4 P45985 2/20 0.38
GSK3B P49841 2/20 0.38
CYP1A2 P05177 1/20 0.38
ALPL P05186 1/20 0.36
MAPK1 P28482 6/20 0.35
NTRK1 P04629 3/20 0.35
HSP90AB1 P08238 1/20 0.35
GPR17 Q13304 1/20 0.35
PPARG P37231 1/20 0.34
NCOA2 Q15596 1/20 0.34
NCOA1 Q15788 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
NCOA3 Q9Y6Q9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23872474 0.77 KDM4E (0.48) SMN1; SMN2MAPTMAP2K4ALPLMAPK1
SCHEMBL23914767 0.76 MAP2K4 (0.51) SMN1; SMN2MAPTMAP2K4GSK3BCYP1A2
SCHEMBL8219414 0.75 SMN1; SMN2 (0.49) SMN1; SMN2MAPTALPLMAPK1PPARG
SCHEMBL155393 0.71 HSP90AB1 (0.46) SMN1; SMN2MAPTHSP90AB1RXFP1
SCHEMBL29324357 0.71 GPR17 (0.35) SMN1; SMN2MAPTMAP2K4ALPLMAPK1
SCHEMBL21801325 0.71 AGBL2 (0.49) SMN1; SMN2MAPTMAPK1HSP90AB1
SCHEMBL23858844 0.69 HCAR2 (0.44) MAP2K4ALPLMAPK1GPR17
SCHEMBL30050008 0.69 HCAR2 (0.44) MAP2K4ALPLMAPK1GPR17
SCHEMBL4300704 0.69 SMN1; SMN2 (0.71) SMN1; SMN2MAPT
SCHEMBL14564361 0.69 SMN1; SMN2 (0.55) SMN1; SMN2MAPTMAP2K4GSK3BCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008040995-A9 INDAZOLES FOR USE AS DPP-IV INHIBITORS PEAKDALE MOLECULAR LTD (GB) 2008-12-31 WO disclosed
WO-2008040995-A1 INDAZOLES FOR USE AS DPP-IV INHIBITORS PEAKDALE MOLECULAR LIMITED (GB) 2008-04-10 WO disclosed