SCHEMBL8205300

SCHEMBL8205300

Cc1cccc(C)c1OC(C)CN(C)CCc1ccc(N)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.40
ADRA2A P08913 1/20 0.37
ADRA2B P18089 1/20 0.37
ADRA2C P18825 1/20 0.37
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
SCN4A P35499 7/20 0.35
LMNA P02545 2/20 0.35
SCN1A P35498 2/20 0.35
KCNH2 Q12809 2/20 0.35
SCN5A Q14524 2/20 0.35
SCN9A Q15858 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2D6 P10635 2/20 0.35
NFKB1 P19838 2/20 0.35
MAOA P21397 2/20 0.35
CYP2C9 P11712 1/20 0.35
TSHR P16473 1/20 0.35
KCNK3 O14649 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8213354 0.82 KCNH2 (0.50) SIGMAR1MEN1KMT2AKCNH2TSHR
SCHEMBL8205331 0.80 KCNH2 (0.52) LMNAKCNH2CYP1A2CYP3A4CYP2D6
SCHEMBL8214024 0.80 SCN8A (0.47) MEN1KMT2ALMNASCN8AAOC3
Hydrochloric Acid SCHEMBL8216124 0.79 KCNH2 (0.51) LMNAKCNH2CYP1A2CYP3A4CYP2D6
SCHEMBL7697582 0.77 KCNH2 (0.52) SIGMAR1SCN4ALMNASCN1AKCNH2
SCHEMBL8203613 0.77 HRH3 (0.43) CYP1A2CYP3A4CYP2C9SCN8A
SCHEMBL7695490 0.74 SCN4A (0.48) SIGMAR1SCN4ALMNASCN1AKCNH2
SCHEMBL7697606 0.74 SCN4A (0.48) SIGMAR1SCN4ALMNASCN1AKCNH2
SCHEMBL7695487 0.74 SCN4A (0.48) SIGMAR1SCN4ALMNASCN1AKCNH2
SCHEMBL9627913 0.71 SIGMAR1 (0.66) SIGMAR1KCNH2CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1037871-A1 NOVEL ANTIARRHYTHMIC COMPOUNDS GYOGYSZERKUTATO INTEZET KFT. (HU) 2000-09-27 EP disclosed
WO-1999029655-A1 NOVEL ANTIARRHYTHMIC COMPOUNDS Gyógyszerkutató Intézet Kft. (HU) 1999-06-17 WO disclosed