SCHEMBL8205331

SCHEMBL8205331

Cc1cccc(C)c1OC(C)CN(C)CCc1ccc(NS(C)(=O)=O)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 8/20 0.52
CACNA1F O60840 1/20 0.52
CHRM2 P08172 1/20 0.52
ACHE P22303 1/20 0.52
AGTR1 P30556 1/20 0.52
DRD3 P35462 1/20 0.52
CACNA1D Q01668 1/20 0.52
CACNA1S Q13698 1/20 0.52
CACNA1C Q13936 1/20 0.52
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
MAPK1 P28482 1/20 0.46
CYP2C19 P33261 1/20 0.46
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8216124 0.99 KCNH2 (0.51) KCNH2CACNA1FCHRM2ACHEAGTR1
Hydrochloric Acid SCHEMBL8216596 0.87 KCNH2 (0.50) KCNH2CACNA1FCHRM2ACHEAGTR1
SCHEMBL6140360 0.87 KCNH2 (0.50) KCNH2CACNA1FCHRM2ACHEAGTR1
SCHEMBL8214024 0.82 SCN8A (0.47) DRD3MAPK1ALDH1A1LMNAHTT
Hydrochloric Acid SCHEMBL8214038 0.81 KCNH2 (0.48) KCNH2CACNA1FCHRM2ACHEAGTR1
SCHEMBL8205300 0.80 SIGMAR1 (0.40) KCNH2CACNA1FCACNA1DCACNA1SCACNA1C
Hydrochloric Acid SCHEMBL8205350 0.80 KCNH2 (0.49) KCNH2CACNA1FCHRM2ACHEAGTR1
Hydrochloric Acid SCHEMBL7702945 0.80 KCNH2 (0.70) KCNH2CACNA1FCHRM2ACHEAGTR1
SCHEMBL8214793 0.80 KCNH2 (0.49) KCNH2KDM4EALDH1A1LMNAHPGD
SCHEMBL8203613 0.79 HRH3 (0.43) CYP1A2CYP3A4CYP2C9MAPK1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1037871-A1 NOVEL ANTIARRHYTHMIC COMPOUNDS GYOGYSZERKUTATO INTEZET KFT. (HU) 2000-09-27 EP claimed
WO-1999029655-A1 NOVEL ANTIARRHYTHMIC COMPOUNDS Gyógyszerkutató Intézet Kft. (HU) 1999-06-17 WO claimed