SCHEMBL8206566

SCHEMBL8206566

Cn1nc(-c2ccccc2)c(-c2cccnc2F)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 4/20 0.41
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HTT P42858 1/20 0.36
HSD17B10 Q99714 1/20 0.36
TOP1 P11387 1/20 0.36
GRM5 P41594 1/20 0.36
NSD3 Q9BZ95 1/20 0.36
FEN1 P39748 1/20 0.35
CTSD P07339 1/20 0.35
BACE1 P56817 1/20 0.35
BACE2 Q9Y5Z0 1/20 0.35
METAP2 P50579 1/20 0.35
CYP11B2 P19099 1/20 0.35
CDK1 P06493 1/20 0.35
CDK4 P11802 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13509078 0.85 DHODH (0.40) DHODHMAOAMAOBPTGS1PTGS2
SCHEMBL13510736 0.85 DHODH (0.40) DHODHMAOAMAOBPTGS1PTGS2
SCHEMBL8214339 0.79 KDM4E (0.43) PTGS1PTGS2KDM4EHTTTOP1
SCHEMBL8205966 0.77 KMT2A (0.48) ALDH1A1KDM4EHTTHSD17B10NSD3
SCHEMBL31051044 0.75 DHODH (0.50) DHODHMAOAMAOBPTGS1PTGS2
SCHEMBL3876408 0.75 DHODH (0.50) DHODHMAOAMAOBPTGS1PTGS2
SCHEMBL28251774 0.75 ALDH1A1 (0.43) ALDH1A1KDM4EHSD17B10NPC1RAB9A
SCHEMBL8212224 0.74 NSD3 (0.41) ALDH1A1KDM4EGRM5NSD3PDE10A
SCHEMBL8215286 0.69 KMT2A (0.41) ALDH1A1KDM4EHTTHSD17B10NSD3
SCHEMBL16200271 0.68 ALDH1A1 (0.40) DHODHMAOAMAOBALDH1A1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021960-A2 TRIAZOLYL MACROCYCLIC HEPATITIS C SERINE PROTEASE INHIBITORS ENANTA PHARMACEUTICALS, INC. (US) 2008-02-21 WO disclosed