SCHEMBL16200271

SCHEMBL16200271

Cc1c(Cl)c(-c2cccnc2F)nn1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
GFER P55789 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
THRB P10828 1/20 0.39
PDE10A Q9Y233 3/20 0.38
CYP11B2 P19099 1/20 0.37
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
BRD4 O60885 2/20 0.35
DHODH Q02127 2/20 0.35
PDE2A O00408 2/20 0.35
PDE4D Q08499 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
MAPT P10636 2/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
ADCY10 Q96PN6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16200388 0.80 THRB (0.45) ALDH1A1GFERNPSR1RXFP1THRB
SCHEMBL16200246 0.79 ALDH1A1 (0.39) ALDH1A1PDE10ACYP11B2BRD4DHODH
SCHEMBL13683013 0.75 THRB (0.42) ALDH1A1GFERNPSR1RXFP1THRB
SCHEMBL13430363 0.73 KDM4E (0.45) ALDH1A1NPSR1THRBPDE10AGAA
SCHEMBL13184428 0.71 SLC34A1 (0.53) ALDH1A1GFERNPSR1RXFP1THRB
SCHEMBL16200197 0.71 CYP11B2 (0.38) CYP11B2DHODHMAPT
SCHEMBL16200063 0.69 ALDH1A1 (0.48) ALDH1A1THRBCYP11B2
SCHEMBL16200060 0.68 THRB (0.52) ALDH1A1NPSR1THRBGAAHPGD
SCHEMBL8206566 0.68 DHODH (0.41) ALDH1A1PDE10ACYP11B2DHODHPDE2A
SCHEMBL16200055 0.67 MAPK14 (0.43) ALDH1A1GFERNPSR1RXFP1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed