SCHEMBL8206848

SCHEMBL8206848

CC(c1ccccc1)N1CCc2cc(NC(=O)c3ccccc3-c3ccc(C(F)(F)F)cc3)ccc2C1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MTTP P55157 18/20 0.56
APOB P04114 9/20 0.56
SMO Q99835 1/20 0.49
KDM4E B2RXH2 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8208880 1.00 MTTP (0.56) MTTPAPOBSMOKDM4E
SCHEMBL8199895 0.91 APOB (0.57) MTTPAPOBSMOKDM4E
SCHEMBL8207411 0.91 MTTP (0.60) MTTPAPOBSMOKDM4E
SCHEMBL4965235 0.87 MTTP (0.60) MTTPAPOBSMOKDM4E
SCHEMBL8208392 0.86 MTTP (0.58) MTTPAPOBSMOKDM4E
SCHEMBL690258 0.84 APOB (0.56) MTTPAPOBSMOKDM4E
SCHEMBL8210365 0.84 MTTP (0.53) MTTPAPOBSMOKDM4E
SCHEMBL6966884 0.84 APOB (0.61) MTTPAPOBSMOKDM4E
SCHEMBL8212442 0.83 APOB (0.54) MTTPAPOBSMOKDM4E
SCHEMBL6966949 0.83 MTTP (0.53) MTTPAPOBSMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6121283-A Apo B-secretion/MTP inhibitory amides PFIZER INC (US) 2000-09-19 US claimed
EP-0944602-A1 APO B-SECRETION/MTP INHIBITORY AMIDES PFIZER INC. (US) 1999-09-29 EP claimed
WO-1998023593-A1 APO B-SECRETION/MTP INHIBITORY AMIDES PFIZER INC. (US) 1998-06-04 WO claimed
US-6121283-A Apo B-secretion/MTP inhibitory amides PFIZER INC (US) 2000-09-19 US disclosed
EP-0944602-A1 APO B-SECRETION/MTP INHIBITORY AMIDES PFIZER INC. (US) 1999-09-29 EP disclosed
WO-1998023593-A1 APO B-SECRETION/MTP INHIBITORY AMIDES PFIZER INC. (US) 1998-06-04 WO disclosed