SCHEMBL6966949

SCHEMBL6966949

C[C@@H](NC(=O)ON1CCc2cc(NC(=O)c3ccccc3-c3ccc(C(F)(F)F)cc3)ccc2C1)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MTTP P55157 19/20 0.53
APOB P04114 9/20 0.53
SMO Q99835 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974830 0.88 MTTP (0.56) MTTPAPOBSMO
SCHEMBL6974648 0.84 MTTP (0.60) MTTPAPOBSMO
SCHEMBL8208880 0.83 MTTP (0.56) MTTPAPOBSMO
SCHEMBL8206848 0.83 MTTP (0.56) MTTPAPOBSMO
SCHEMBL6970130 0.82 SMO (0.54) MTTPAPOBSMO
SCHEMBL6973182 0.82 MTTP (0.52) MTTPAPOBSMO
SCHEMBL8199895 0.81 APOB (0.57) MTTPAPOBSMO
SCHEMBL8207411 0.81 MTTP (0.60) MTTPAPOBSMO
SCHEMBL690258 0.80 APOB (0.56) MTTPAPOBSMO
SCHEMBL4965235 0.79 MTTP (0.60) MTTPAPOBSMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832069-B1 BIPHENYL-2-CARBOXYLIC ACID-TETRAHYDRO-ISOQUINOLIN-6-YL AMIDE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS INHIBITORS OF MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN AND/OR APOLIPOPROTEIN B (Apo B) SECRETION PFIZER (US) 2003-03-05 EP claimed