SCHEMBL8207645

SCHEMBL8207645

Cc1ccc(Br)c(C(=O)N2C[C@H]3C[C@H]3[C@H]2C)c1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.35
HPGD P15428 2/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
HTT P42858 2/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HCRTR1 O43613 6/20 0.34
HCRTR2 O43614 6/20 0.34
POLB P06746 2/20 0.34
CPS1 P31327 2/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
TP53 P04637 1/20 0.32
F2R P25116 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
PKM P14618 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8212395 0.90 ALDH1A1 (0.38) ALDH1A1HPGDMEN1KMT2AHTT
SCHEMBL2931508 0.84 POLB (0.38) ALDH1A1HPGDMEN1KMT2AHTT
SCHEMBL2931509 0.83 HTR2A (0.35) ALDH1A1HPGDMEN1KMT2AHTT
SCHEMBL8205452 0.76 MGLL (0.40) ALDH1A1HPGDHTTHCRTR1HCRTR2
SCHEMBL2931793 0.73 POLB (0.38) ALDH1A1HPGDMEN1KMT2AHTT
SCHEMBL2931198 0.73 HTR2A (0.38) ALDH1A1HPGDMEN1KMT2AHTT
SCHEMBL2931197 0.73 HTR2A (0.38) ALDH1A1HPGDMEN1KMT2AHTT
SCHEMBL3460327 0.67 HCRTR1 (0.45) HCRTR1HCRTR2
SCHEMBL2927512 0.67 CYP46A1 (0.41) HCRTR1HCRTR2POLB
SCHEMBL16277556 0.67 HCRTR1 (0.47) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079690-B1 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-09-15 EP disclosed
WO-2008038251-A2 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2008-04-03 WO disclosed