SCHEMBL8207786

SCHEMBL8207786

COC(=O)CCN1CCC(=C2c3ccn(C)c3CCn3ncnc32)CC1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.33
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CACNA1C Q13936 1/20 0.31
HTR1A P08908 3/20 0.31
DRD2 P14416 3/20 0.31
HTR2A P28223 3/20 0.31
NOTUM Q6P988 1/20 0.30
KDM1A O60341 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL7138914 0.82 KDM4E (0.40) HRH1KDM4EALDH1A1CACNA1CHTR1A
SCHEMBL7140680 0.81 PTAFR (0.40) HRH1ALDH1A1DRD2
SCHEMBL8207783 0.81 HRH3 (0.46) HRH1HTR1A
SCHEMBL8208865 0.81 HRH1 (0.52) HRH1ALDH1A1HTR1ADRD2HTR2A
SCHEMBL8212560 0.78 HRH1 (0.40) HRH1HTR1ADRD2HTR2A
Water SCHEMBL6994538 0.74 HRH1 (0.62) HRH1SMN1; SMN2HTR2A
SCHEMBL7893060 0.70 HRH1 (0.44) HRH1SMN1; SMN2KDM4EALDH1A1CACNA1C
SCHEMBL6991699 0.70 HRH1 (0.68) HRH1HTR1ADRD2HTR2A
Water SCHEMBL9383772 0.69 HRH1 (0.57) HRH1
SCHEMBL7895280 0.68 HRH1 (0.42) HRH1SMN1; SMN2KDM4EALDH1A1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0675889-B1 ANTIALLERGIC TRIAZOLO(PYRROLO, THIENO OR FURANO)AZEPINE DERIVATIVES JANSSEN PHARMACEUTICA NV (BE) 2000-07-05 EP disclosed
US-5595988-A Triazolo(pyrrolo, thieno or furano)azepine derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1997-01-21 US disclosed