SCHEMBL8207983

SCHEMBL8207983

Cc1ccc2c3c(c4ccccc4cc13)C(=O)NC2=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.50
MAPT P10636 4/20 0.40
NPSR1 Q6W5P4 2/20 0.40
CYP1A2 P05177 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
RGS12 O14924 1/20 0.40
USP2 O75604 1/20 0.40
POLB P06746 1/20 0.40
CYP3A4 P08684 1/20 0.40
THRB P10828 1/20 0.40
CYP2C9 P11712 1/20 0.40
APEX1 P27695 1/20 0.40
CASP1 P29466 1/20 0.40
BRCA1 P38398 1/20 0.40
MTOR P42345 1/20 0.40
RECQL P46063 1/20 0.40
BLM P54132 1/20 0.40
CASP7 P55210 1/20 0.40
GNAI1 P63096 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18676726 0.80 CES1 (0.61) MAPTNPSR1CYP1A2MEN1KMT2A
SCHEMBL3079295 0.78 CES1 (0.63) PARP1MAPTNPSR1CYP1A2MEN1
SCHEMBL31241414 0.78 CES1 (0.63) PARP1MAPTNPSR1CYP1A2MEN1
SCHEMBL26507159 0.78 TYMS (0.41) MAPTCYP1A2KMT2ATDP1KDM4E
SCHEMBL6405656 0.76 PARP1 (0.53) PARP1MAPTNPSR1CYP1A2MEN1
SCHEMBL1889878 0.76 PARP1 (0.55) PARP1MAPTNPSR1CYP1A2MEN1
SCHEMBL9968963 0.74 MEN1 (0.62) PARP1MAPTNPSR1CYP1A2MEN1
SCHEMBL7278240 0.73 GSK3B (0.44) PARP1MAPTNPSR1MEN1KMT2A
SCHEMBL57037 0.72 DNMT1 (0.53) PARP1MAPTNPSR1CYP1A2MEN1
SCHEMBL1654813 0.72 ALOX5 (0.51) PARP1MEN1KMT2ARECQLTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008033891-A2 AZONAFIDE DERIVED TUMOR AND CANCER TARGETING COMPOUNDS GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2008-03-20 WO disclosed