SCHEMBL8208041

SCHEMBL8208041

C=CCOc1ccc(C[C@H](BOCN)C(=O)N[C@@H](CC(C)C)C(=O)OC)cc1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IL1RN P18510 3/20 0.45
ERAP2 Q6P179 3/20 0.45
ERAP1 Q9NZ08 3/20 0.45
TAS1R3 Q7RTX0 6/20 0.41
TAS1R1 Q7RTX1 6/20 0.41
BIRC2 Q13490 1/20 0.41
MMP1 P03956 4/20 0.39
MMP3 P08254 2/20 0.39
MMP9 P14780 2/20 0.39
ADAM17 P78536 1/20 0.39
MMP2 P08253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12943098 0.93 IL1RN (0.45) IL1RNERAP2ERAP1TAS1R3TAS1R1
SCHEMBL12943165 0.92 IL1RN (0.44) IL1RNERAP2ERAP1MMP1MMP3
SCHEMBL8208994 0.92 MME (0.42) MMP1MMP3MMP9ADAM17MMP2
SCHEMBL8202825 0.92 PTPN1 (0.44) IL1RNERAP2ERAP1MMP1MMP3
SCHEMBL8211378 0.91 IL1RN (0.47) IL1RNERAP2ERAP1TAS1R3TAS1R1
SCHEMBL12943096 0.91 IL1RN (0.43) IL1RNERAP2ERAP1TAS1R3TAS1R1
SCHEMBL12907549 0.89 IL1RN (0.46) IL1RNERAP2ERAP1TAS1R3TAS1R1
SCHEMBL8201294 0.88 PTPN1 (0.39) IL1RNERAP2ERAP1MMP1MMP3
SCHEMBL8209110 0.86 PTPN1 (0.38) IL1RNERAP2ERAP1MMP1MMP3
SCHEMBL12943214 0.86 CTSB (0.38) MMP1MMP3MMP9MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008048121-A2 MACROCYCLIC CYSTEINE PROTEASE INHIBITORS AND COMPOSITIONS THEREOF LINCOLN UNIVERSITY (NZ) 2008-04-24 WO disclosed