SCHEMBL8209110

SCHEMBL8209110

C=CCOC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](BOCN)Cc1ccc(OCC=C)cc1)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.38
IL1RN P18510 2/20 0.38
ERAP2 Q6P179 2/20 0.38
ERAP1 Q9NZ08 2/20 0.38
OPRM1 P35372 4/20 0.37
OPRK1 P41145 4/20 0.37
MMP1 P03956 2/20 0.36
MME P08473 1/20 0.36
NPY1R P25929 1/20 0.35
NPY2R P49146 1/20 0.35
NPY4R P50391 1/20 0.35
ITGB3 P05106 1/20 0.35
ITGA2B P08514 1/20 0.35
MMP2 P08253 1/20 0.35
MMP3 P08254 1/20 0.35
MMP9 P14780 1/20 0.35
KLKB1 P03952 1/20 0.35
PSMB5 P28074 1/20 0.35
PSMB2 P49721 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12943098 0.93 IL1RN (0.45) PTPN1IL1RNERAP2ERAP1OPRM1
SCHEMBL8208994 0.92 MME (0.42) PTPN1MMP1MMEITGB3ITGA2B
SCHEMBL8201294 0.90 PTPN1 (0.39) PTPN1IL1RNERAP2ERAP1OPRM1
SCHEMBL8202825 0.87 PTPN1 (0.44) PTPN1IL1RNERAP2ERAP1OPRM1
SCHEMBL8208041 0.86 IL1RN (0.45) IL1RNERAP2ERAP1MMP1MMP2
SCHEMBL12943165 0.86 IL1RN (0.44) PTPN1IL1RNERAP2ERAP1OPRM1
SCHEMBL12943085 0.84 ITGB3 (0.44) IL1RNERAP2ERAP1MMP1MME
SCHEMBL12943096 0.83 IL1RN (0.43) PTPN1IL1RNERAP2ERAP1OPRM1
SCHEMBL12943214 0.82 CTSB (0.38) MMP1MMP2MMP3MMP9
SCHEMBL8208453 0.81 ITGB3 (0.36) MMP1MMEITGB3ITGA2BMMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008048121-A2 MACROCYCLIC CYSTEINE PROTEASE INHIBITORS AND COMPOSITIONS THEREOF LINCOLN UNIVERSITY (NZ) 2008-04-24 WO disclosed