SCHEMBL8208739

SCHEMBL8208739

Nc1nc2[nH]cnc2c(=O)n1Cc1ccc(-c2ccccc2)s1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNP P00491 3/20 0.40
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
CYP2E1 P05181 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2A6 P11509 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2B6 P20813 1/20 0.39
CYP2C19 P33261 1/20 0.39
KLKB1 P03952 2/20 0.37
KLK1 P06870 2/20 0.37
RAB9A P51151 3/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
HPGD P15428 1/20 0.35
NPC1 O15118 1/20 0.35
MAPT P10636 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
APP P05067 1/20 0.34
BACE1 P56817 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8208746 0.82 PNP (0.45) PNPCYP11B1CYP11B2CYP2E1CYP3A4
SCHEMBL9434507 0.81 PNP (0.35) PNPALDH1A1HPGDMAPTSMN1; SMN2
SCHEMBL3300181 0.81 PNP (0.35) PNP
SCHEMBL4963405 0.81 MGMT (0.35) PNPALDH1A1MAPTKDM4E
SCHEMBL18247 0.81 PNP (0.59) PNPALDH1A1MAPTKDM4E
SCHEMBL4966163 0.80 ADRA1D (0.39) PNPCYP2A6
SCHEMBL1980958 0.80 PNP (0.57) PNPALDH1A1MAPTKDM4E
SCHEMBL4962851 0.79 PNP (0.53) PNPCYP3A4CYP2C9CYP2C19ALDH1A1
Hydrochloric Acid SCHEMBL17186370 0.78 PNP (0.52) PNPCYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL1938284 0.76 KMT2A (0.42) PNPALDH1A1LMNAMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6096724-A O(6)-ALKYLGUANINE-DNA ALKYLTRANSFERASE (ATASE) ENZYME INHIBITORS CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2000-08-01 US disclosed