SCHEMBL8208741

SCHEMBL8208741

COc1cnc(/C=C/C(=O)c2ccccc2)cc1OCc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.57
ALDH1A1 P00352 1/20 0.57
THRB P10828 1/20 0.57
NPC1 O15118 3/20 0.52
RAB9A P51151 3/20 0.52
MAPT P10636 2/20 0.52
MAOB P27338 1/20 0.52
MRGPRX4 Q96LA9 1/20 0.51
PTPN1 P18031 1/20 0.51
ATM Q13315 1/20 0.50
PTGER4 P35408 1/20 0.49
PTGER2 P43116 1/20 0.49
APP P05067 2/20 0.49
HPGD P15428 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
BCHE P06276 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
SMPD1 P17405 1/20 0.48
HDAC1 Q13547 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8208745 1.00 LMNA (0.57) LMNAALDH1A1THRBNPC1RAB9A
SCHEMBL8219209 0.89 NPC1 (0.60) LMNAALDH1A1NPC1RAB9AMAPT
SCHEMBL8219212 0.89 NPC1 (0.60) LMNAALDH1A1NPC1RAB9AMAPT
SCHEMBL8209030 0.87 NPC1 (0.53) LMNAALDH1A1NPC1RAB9AMAPT
SCHEMBL8220667 0.87 NPC1 (0.53) LMNAALDH1A1NPC1RAB9AMAPT
SCHEMBL8220517 0.86 NPC1 (0.52) LMNAALDH1A1THRBNPC1RAB9A
SCHEMBL8220519 0.86 NPC1 (0.52) LMNAALDH1A1THRBNPC1RAB9A
SCHEMBL8211779 0.85 NPC1 (0.54) LMNAALDH1A1NPC1RAB9AMAPT
SCHEMBL8211777 0.85 NPC1 (0.54) LMNAALDH1A1NPC1RAB9AMAPT
SCHEMBL8216223 0.84 NPC1 (0.50) LMNAALDH1A1NPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6046218-A 4,5-DIMETHOXY-2-(3-OXO-3-PHENYL-1-PROPENYL)PYRIDINE USED TO CURE THE DISEASES PRODUCED BY CYTOKINE SS PHARMACEUTICAL CO., LTD. (JP) 2000-04-04 US disclosed
EP-0838457-A1 NOVEL PYRIDINE DERIVATIVES AND MEDICINES CONTAINING THE SAME AS ACTIVE INGREDIENT SS Pharmaceutical Co., Ltd. (JP) 1998-04-29 EP disclosed