SCHEMBL8209031

SCHEMBL8209031

COc1cccc2c1CCN2Cc1cnc[nH]1

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.61
NOTUM Q6P988 1/20 0.44
HDAC1 Q13547 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
FNTA P49354 8/20 0.43
FNTB P49356 8/20 0.43
PKM P14618 1/20 0.41
CYP11B2 P19099 1/20 0.40
HRH4 Q9H3N8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8205622 0.93 TAAR1 (0.62) TAAR1NOTUMHDAC1HDAC6FNTA
SCHEMBL8203976 0.85 TAAR1 (0.64) TAAR1NOTUMFNTAFNTB
SCHEMBL8203733 0.82 TAAR1 (0.59) TAAR1HDAC1HDAC6FNTAFNTB
SCHEMBL8203453 0.82 TAAR1 (0.64) TAAR1NOTUMFNTAFNTB
SCHEMBL12993144 0.81 TAAR1 (0.60) TAAR1FNTAFNTB
SCHEMBL12993166 0.78 TAAR1 (0.58) TAAR1FNTAFNTBHRH4
SCHEMBL1734486 0.78 ADRA2A (0.44) TAAR1NOTUMHDAC1HDAC6FNTA
SCHEMBL508524 0.76 TAAR1 (1.00) TAAR1FNTAFNTB
SCHEMBL11304976 0.76 HTR6 (0.62) NOTUMHDAC1HDAC6
SCHEMBL12993223 0.76 TAAR1 (0.41) TAAR1FNTAFNTBPKMCYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008058867-A2 SUBSTITUTED 4-IMIDAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2008-05-22 WO disclosed