SCHEMBL8209801

SCHEMBL8209801

COc1ccc(C=Cc2ccc3[nH]cc(C4CCN(C)CC4)c3c2)cc1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 7/20 0.58
HTR1B P28222 7/20 0.58
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2D6 P10635 1/20 0.58
CYP2C9 P11712 1/20 0.58
THPO P40225 1/20 0.58
APP P05067 2/20 0.53
MAPT P10636 1/20 0.53
BLM P54132 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
HTR1A P08908 5/20 0.51
HTR1F P30939 2/20 0.51
CCR2 P41597 2/20 0.49
SLC6A4 P31645 3/20 0.49
MTNR1A P48039 1/20 0.48
MTNR1B P49286 1/20 0.48
DRD2 P14416 1/20 0.48
HTR2A P28223 1/20 0.48
HTR7 P34969 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8205314 0.87 HTR1D (0.62) HTR1DHTR1BCYP1A2CYP3A4CYP2D6
SCHEMBL8205310 0.87 HTR1D (0.62) HTR1DHTR1BCYP1A2CYP3A4CYP2D6
SCHEMBL7710792 0.87 HTR1D (0.67) HTR1DHTR1BCYP1A2CYP3A4CYP2D6
SCHEMBL8187195 0.86 HTR1D (0.60) HTR1DHTR1BCYP1A2CYP3A4CYP2D6
SCHEMBL7020706 0.85 HTR1D (0.62) HTR1DHTR1BCYP1A2CYP3A4CYP2D6
SCHEMBL7489712 0.82 HTR1D (0.58) HTR1DHTR1BCYP1A2CYP3A4CYP2D6
SCHEMBL8185092 0.81 HTR1D (0.57) HTR1DHTR1BCYP1A2CYP3A4CYP2D6
SCHEMBL7013891 0.81 HTR1D (0.66) HTR1DHTR1BCYP1A2CYP3A4CYP2D6
SCHEMBL7478910 0.80 CYP1A2 (0.59) HTR1DHTR1BCYP1A2CYP3A4CYP2D6
SCHEMBL25072243 0.80 MTNR1A (0.65) HTR1DHTR1BCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000000490-A2 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 2000-01-06 WO disclosed