SCHEMBL8212907

SCHEMBL8212907

COc1cccc(-c2ccc(C(=O)OC(C)(C)C)c(Cc3cc(F)ccc3F)n2)c1F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.37
MTNR1B P49286 1/20 0.37
PLA2G2A P14555 1/20 0.36
TRPV3 Q8NET8 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
FYN P06241 1/20 0.35
DHODH Q02127 2/20 0.35
CNR1 P21554 2/20 0.34
AAK1 Q2M2I8 1/20 0.34
MMP2 P08253 2/20 0.34
MMP12 P39900 2/20 0.34
MMP1 P03956 1/20 0.34
MMP9 P14780 1/20 0.34
CCNT1 O60563 1/20 0.34
CDK9 P50750 1/20 0.34
GUCY1A1 Q02108 1/20 0.34
GUCY1B1 Q02153 1/20 0.34
KCNH2 Q12809 1/20 0.34
HTR2C P28335 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3747145 0.83 CD274 (0.38) ADORA2AADORA1FYNDHODHCCNT1
SCHEMBL3763504 0.79 AAK1 (0.39) ADORA2AADORA1FYNDHODHAAK1
SCHEMBL8218291 0.78 TRPV3 (0.46) TRPV3GUCY1A1GUCY1B1KCNH2
SCHEMBL8214930 0.72 DHODH (0.40) TRPV3ADORA2AADORA1DHODH
SCHEMBL3749641 0.71 DHODH (0.45) ADORA2AADORA1DHODHCCNT1CDK9
SCHEMBL23943222 0.67 CD274 (0.46) PLA2G2AADORA2AADORA1FYNDHODH
SCHEMBL8214581 0.67 ERN1 (0.33) TRPV3
SCHEMBL23925778 0.67 CD274 (0.46) ADORA2AADORA1FYNDHODHCCNT1
SCHEMBL3757598 0.67 ADORA2A (0.39) ADORA2AADORA1FYNDHODHGPBAR1
SCHEMBL3755649 0.66 DHODH (0.47) ADORA2AADORA1DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008031501-A2 2-PHENOXY NICOTINE ACID DERIVATIVE AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-03-20 WO disclosed