SCHEMBL8214930

SCHEMBL8214930

O=C(O)c1ccc(-c2ccccc2F)nc1Cc1cc(F)ccc1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 5/20 0.40
TRPV3 Q8NET8 1/20 0.40
KMO O15229 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
CTSA P10619 2/20 0.39
ACMSD Q8TDX5 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CASP3 P42574 1/20 0.39
SENP8 Q96LD8 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SENP6 Q9GZR1 1/20 0.39
PTGER1 P34995 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA2B P29275 1/20 0.38
ADORA1 P30542 1/20 0.38
SIRT5 Q9NXA8 1/20 0.37
DHFR P00374 1/20 0.37
ALKBH5 Q6P6C2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8218291 0.81 TRPV3 (0.46) TRPV3CTSA
SCHEMBL8211093 0.73 KDM4E (0.39) DHODHTRPV3KMOCTSAPTGER1
SCHEMBL8202794 0.73 MPL (0.38) DHODHTRPV3BRS3KDM4EALDH1A1
SCHEMBL8212907 0.72 MTNR1A (0.37) DHODHTRPV3ADORA2AADORA1
SCHEMBL11823508 0.72 DCLRE1B (0.46) KDM4EALDH1A1HPGD
SCHEMBL21811216 0.71 PARP1 (0.48) DHODHNPC1RAB9AACMSDSIRT5
SCHEMBL8214581 0.71 ERN1 (0.33) TRPV3L3MBTL1CASP3SENP8SENP7
SCHEMBL8214589 0.70 EIF4E (0.43) DHODHTRPV3KMOCTSAKDM4E
SCHEMBL31490593 0.69 DHODH (0.69) DHODHNPC1RAB9ADHFRALKBH5
SCHEMBL31212334 0.69 PARP1 (0.46) DHODHNPC1RAB9AACMSDSIRT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008031501-A2 2-PHENOXY NICOTINE ACID DERIVATIVE AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-03-20 WO disclosed