SCHEMBL8212975

SCHEMBL8212975

C=CC[C@H](C)COC(N)=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.39
ALOX15 P16050 1/20 0.38
CHRNB2 P17787 2/20 0.36
CHRNA4 P43681 2/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CYP1A2 P05177 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
CYP2D6 P10635 1/20 0.35
PKM P14618 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
LMNA P02545 3/20 0.33
KDM4E B2RXH2 1/20 0.33
CHRM2 P08172 3/20 0.32
CHRM4 P08173 3/20 0.32
CHRM5 P08912 3/20 0.32
CHRM1 P11229 3/20 0.32
CHRM3 P20309 3/20 0.32
GRIK1 P39086 2/20 0.32
GRIK2 Q13002 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8221276 1.00 TSHR (0.39) TSHRALOX15CHRNB2CHRNA4CHRNB4
SCHEMBL28773870 1.00 TSHR (0.39) TSHRALOX15CHRNB2CHRNA4CHRNB4
SCHEMBL7686788 0.82 TSHR (0.41) TSHRSMN1; SMN2LMNATDP1MAPT
SCHEMBL9541479 0.82 TSHR (0.41) TSHRSMN1; SMN2LMNAGRIK1GRIK2
SCHEMBL9541472 0.82 TSHR (0.41) TSHRSMN1; SMN2LMNATDP1MAPT
SCHEMBL8221270 0.81 TSHR (0.41) TSHRALOX15CHRNB2CHRNA4CHRNB4
SCHEMBL30357063 0.80 ALOX15 (0.50) TSHRALOX15CHRNB2CHRNA4CHRNB4
SCHEMBL19442152 0.75
SCHEMBL28725124 0.74 GAA (0.52) TSHRSMN1; SMN2NPSR1LMNATDP1
SCHEMBL28725161 0.74 TSHR (0.35) TSHRGRIK1GRIK2CYP2C19MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008057208-A2 HCV NS3 PROTEASE INHIBITORS MERCK & CO., INC. (US) 2008-05-15 WO disclosed