SCHEMBL8213428

SCHEMBL8213428

N[C@@H](CC(=O)O)C(=O)Nc1ccccc1C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.57
RECQL P46063 1/20 0.57
LTA4H P09960 2/20 0.52
CFD P00746 1/20 0.51
HCAR2 Q8TDS4 4/20 0.51
KMT2A Q03164 5/20 0.49
MAPT P10636 1/20 0.49
CTSK P43235 1/20 0.49
ALDH1A1 P00352 2/20 0.47
HPGD P15428 1/20 0.47
HSD17B10 Q99714 1/20 0.47
MEN1 O00255 3/20 0.47
CASR P41180 1/20 0.47
LMNA P02545 1/20 0.47
PKM P14618 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
DHODH Q02127 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Potassium Ion SCHEMBL8214287 0.87 LTA4H (0.49) KDM4ERECQLLTA4HCFDHCAR2
SCHEMBL10796640 0.85 LARS1 (0.52) KDM4ECFDHCAR2KMT2AMAPT
Hydrochloric Acid SCHEMBL10799048 0.84 LARS1 (0.51) KDM4ECFDHCAR2KMT2AMAPT
SCHEMBL32666130 0.83 HCAR2 (0.50) KDM4ERECQLLTA4HCFDHCAR2
SCHEMBL6046896 0.83 HDAC1 (0.51) LTA4H
SCHEMBL8171158 0.83 GAA (0.57) KDM4ELTA4HKMT2AMAPTHPGD
SCHEMBL7146676 0.81 HCAR2 (0.44) KDM4ERECQLCFDHCAR2KMT2A
SCHEMBL7146679 0.81 HCAR2 (0.44) KDM4ERECQLCFDHCAR2KMT2A
SCHEMBL8037232 0.79 LTA4H (0.47) KDM4ERECQLLTA4HKMT2AMEN1
SCHEMBL27295439 0.79 KDM4E (0.57) KDM4ELTA4HKMT2AMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6015792-A Specific eatable taste modifiers BIORESEARCH, INC. (US) 2000-01-18 US claimed
US-5631038-A COMPOUNDS (TASTANDS) TO REDUCE OR ELIMINATE A BITTER OR METALLIC TASTE ARE ADDED TO FOODS CONTAINING SODIUM CHLORIDE BIORESEARCH, INC. (US) 1997-05-20 US claimed
EP-0661932-A4 SPECIFIC EATABLE TASTE MODIFIERS. BIORESEARCH INC (US) 1996-06-05 EP claimed
EP-0661932-A1 SPECIFIC EATABLE TASTE MODIFIERS BIORESEARCH, INC. (US) 1995-07-12 EP claimed
WO-1993010677-A1 SPECIFIC EATABLE TASTE MODIFIERS BIORESEARCH, INC. (US) 1993-06-10 WO claimed
US-6015792-A Specific eatable taste modifiers BIORESEARCH, INC. (US) 2000-01-18 US disclosed
US-6008250-A Specific eatable taste modifiers BIORESEARCH, INC. (US) 1999-12-28 US disclosed
US-5866608-A AROMATIC COMPOUNDS BIORESEARCH, INC. (US) 1999-02-02 US disclosed
US-5703053-A TASTELESS INGESTIBLE COMPOUNDS WHICH REDUCE OR ELIMINATE UNDESIRABLE TASTES IN EATABLES BIORESEARCH, INC. (US) 1997-12-30 US disclosed
US-5700792-A Specific eatable taste modifiers BIORESEARCH, INC. (US) 1997-12-23 US disclosed
US-5665755-A NAPHTHO(1,2-D)IMIDAZOLE-5-SULFONATES (TASTANDS) USED TO REDUCE BITTER OR METALLIC TASTES; FOODS, DRUGS, ARTIFICIAL SWEETENERS; POTASSIUM CHLORIDE BIORESEARCH INC. (US) 1997-09-09 US disclosed
US-5654311-A TASTANDS OF PYRIMIDINE DERIVATIVES, E.G. OROTIC ACID, TO REDUCE OR ELIMINATE A BITTER OR METALLIC TASTE; FOODS; DRUGS; SWEETENERS; POTASSIUM CHLORIDE BIORESEARCH INC. (US) 1997-08-05 US disclosed
US-5631038-A COMPOUNDS (TASTANDS) TO REDUCE OR ELIMINATE A BITTER OR METALLIC TASTE ARE ADDED TO FOODS CONTAINING SODIUM CHLORIDE BIORESEARCH, INC. (US) 1997-05-20 US disclosed
US-5631294-A PHENOXY- OR PHENYL-ALKANOIC ACIDS BIORESEARCH, INC. (US) 1997-05-20 US disclosed
US-5631295-A 2-(4-METHOXYPHENOXY)PROPIONIC ACID, TAURINE, ASPARTYLPHENYL ALANINE, ASPARTYLTYROSINE AND DIHYDROXYBENZOIC ACID BIORESEARCH, INC. (US) 1997-05-20 US disclosed
US-5631240-A KETONE BIORESEARCH, INC. (US) 1997-05-20 US disclosed
US-5631299-A TAURINE OR AN ACCEPTABLE SALT (A TASTAND) TO REDUCE OR ELIMINATE A BITTER OR METALLIC TASTE; FOODS; DRUGS; SWEETENERS; POTASSIUM CHLORIDE BIORESEARCH, INC. (US) 1997-05-20 US disclosed
EP-0661932-A4 SPECIFIC EATABLE TASTE MODIFIERS. BIORESEARCH INC (US) 1996-06-05 EP disclosed
EP-0661932-A1 SPECIFIC EATABLE TASTE MODIFIERS BIORESEARCH, INC. (US) 1995-07-12 EP disclosed
WO-1993010677-A1 SPECIFIC EATABLE TASTE MODIFIERS BIORESEARCH, INC. (US) 1993-06-10 WO disclosed