SCHEMBL8213641

SCHEMBL8213641

COC(=O)[C@@H]1COC/C=C/COc2ccc(cc2)C[C@H](BOCN)C(=O)N[C@@H](C(C)C)C(=O)N1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CAPN2 P17655 2/20 0.34
MMP2 P08253 8/20 0.33
MMP7 P09237 8/20 0.33
MMP3 P08254 7/20 0.33
F2 P00734 2/20 0.33
F10 P00742 2/20 0.33
PLG P00747 2/20 0.33
KLKB1 P03952 2/20 0.33
MMP9 P14780 2/20 0.33
PROC P04070 1/20 0.33
MMP12 P39900 1/20 0.33
MMP13 P45452 1/20 0.33
MMP1 P03956 6/20 0.33
ADAM17 P78536 2/20 0.33
ITGB1 P05556 1/20 0.32
ITGA2 P17301 1/20 0.32
CPB2 Q96IY4 3/20 0.32
NTSR1 P30989 1/20 0.32
MCL1 Q07820 1/20 0.32
KRAS P01116 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8208869 0.92 F2 (0.35) CAPN2MMP2MMP7MMP3F2
SCHEMBL8211181 0.92 F2 (0.35) CAPN2MMP2MMP7MMP3F2
SCHEMBL12943278 0.89 TMPRSS2 (0.39) CAPN2MMP2MMP7MMP3F2
SCHEMBL8201392 0.89 TMPRSS2 (0.39) CAPN2MMP2MMP7MMP3F2
SCHEMBL8209145 0.89 CPB2 (0.42) CAPN2MMP2MMP7MMP3MMP9
SCHEMBL12943111 0.87 CAPN2 (0.36) CAPN2MMP2MMP7MMP3F2
SCHEMBL8206145 0.85 MMP2 (0.44) CAPN2MMP2MMP7MMP3MMP9
SCHEMBL8213651 0.84 CAPN2 (0.46) CAPN2MMP2MMP7MMP3MMP9
SCHEMBL15869971 0.78 CAPN2 (0.35) CAPN2MMP2MMP7MMP3F2
SCHEMBL12943279 0.78 MMP2 (0.44) CAPN2MMP2MMP7MMP3MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008048121-A2 MACROCYCLIC CYSTEINE PROTEASE INHIBITORS AND COMPOSITIONS THEREOF LINCOLN UNIVERSITY (NZ) 2008-04-24 WO disclosed