3,4-Dihydroxyphenylacetic Acid

3,4-Dihydroxyphenylacetic Acid

SCHEMBL8214147

O=C(O)Cc1ccc(O)c(O)c1.[NaH]

nearest known ligand 0.96

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 5/20 0.96
KDM4E B2RXH2 5/20 0.96
TDP1 Q9NUW8 4/20 0.96
HSD17B10 Q99714 4/20 0.96
MAPT P10636 4/20 0.96
HPGD P15428 3/20 0.96
TSHR P16473 2/20 0.96
NFKB1 P19838 2/20 0.96
HIF1A Q16665 2/20 0.96
POLB P06746 2/20 0.96
APEX1 P27695 2/20 0.96
BLM P54132 2/20 0.96
PMP22 Q01453 2/20 0.96
RGS12 O14924 1/20 0.96
LMNA P02545 1/20 0.96
THPO P40225 1/20 0.96
GNAI1 P63096 1/20 0.96
CA2 P00918 3/20 0.66
ALDH1A1 P00352 4/20 0.59
CAMK2A Q9UQM7 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
3,4-Dihydroxyphenylacetic Acid SCHEMBL29382155 0.98 GAA (1.00) GAAKDM4ETDP1HSD17B10MAPT
3,4-Dihydroxyphenylacetic Acid SCHEMBL36348 0.98 GAA (1.00) GAAKDM4ETDP1HSD17B10MAPT
3,4-Dihydroxyphenylacetic Acid SCHEMBL8214151 0.96 GAA (0.96) GAAKDM4ETDP1HSD17B10MAPT
3,4-Dihydroxyphenylacetic Acid SCHEMBL18338957 0.90 GAA (0.85) GAAKDM4ETDP1HSD17B10MAPT
3,4-Dihydroxyphenylacetic Acid SCHEMBL21381267 0.90 GAA (0.85) GAAKDM4ETDP1HSD17B10MAPT
3,4-Dihydroxyphenylacetic Acid SCHEMBL175566 0.87 TDP1 (0.79) GAAKDM4ETDP1HSD17B10MAPT
3,4-Dihydroxyphenylacetic Acid SCHEMBL29246309 0.85 GAA (0.76) GAAKDM4ETDP1HSD17B10MAPT
3,4-Dihydroxyphenylacetic Acid SCHEMBL8565392 0.85 GAA (0.76) GAAKDM4ETDP1HSD17B10MAPT
SCHEMBL2050404 0.83 GAA (0.73) GAAKDM4ETDP1HSD17B10MAPT
SCHEMBL15499982 0.83 GAA (0.73) GAAKDM4ETDP1HSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 33 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6015792-A Specific eatable taste modifiers BIORESEARCH, INC. (US) 2000-01-18 US disclosed
US-6008250-A Specific eatable taste modifiers BIORESEARCH, INC. (US) 1999-12-28 US disclosed
US-5866608-A AROMATIC COMPOUNDS BIORESEARCH, INC. (US) 1999-02-02 US disclosed
US-5703053-A TASTELESS INGESTIBLE COMPOUNDS WHICH REDUCE OR ELIMINATE UNDESIRABLE TASTES IN EATABLES BIORESEARCH, INC. (US) 1997-12-30 US disclosed
US-5700792-A Specific eatable taste modifiers BIORESEARCH, INC. (US) 1997-12-23 US disclosed
US-5665755-A NAPHTHO(1,2-D)IMIDAZOLE-5-SULFONATES (TASTANDS) USED TO REDUCE BITTER OR METALLIC TASTES; FOODS, DRUGS, ARTIFICIAL SWEETENERS; POTASSIUM CHLORIDE BIORESEARCH INC. (US) 1997-09-09 US disclosed
US-5654311-A TASTANDS OF PYRIMIDINE DERIVATIVES, E.G. OROTIC ACID, TO REDUCE OR ELIMINATE A BITTER OR METALLIC TASTE; FOODS; DRUGS; SWEETENERS; POTASSIUM CHLORIDE BIORESEARCH INC. (US) 1997-08-05 US disclosed
US-5650403-A PURINE-BASED COMPOUNDS (TASTANDS, E.G. IOSINE, GUANOSINE AND XANTHINE-5'-PHOSPHATE) USED TO REDUCE OR ELIMINATE A BITTER OR METALLIC TASTE; FOODS; DRUGS; ARTIFICIAL SWEETENERS; POTASSIUM CHLORIDE BIORESEARCH, INC. (US) 1997-07-22 US disclosed
US-5646122-A COMPOUNDS (TASTANDS, E.G. A DIPEPTIDE CONTAINING TAURINE AND/OR ALANINE) USED TO REDUCE OR ELIMINATE A BITTER OR METALLIC TASTE; FOODS; DRUGS; ARTIFICIAL SWEETENERS; POTASSIUM CHLORIDE BIORESEARCH, INC. (US) 1997-07-08 US disclosed
US-5643941-A PYRAN, THIOPYRAN AND CYCLOHEXANE DERIVATIVES (E.G. GLYCOSIDES AND INOSITOL, QUERCITOL) TO REDUCE OR ELIMINATE A BITTER OR METALLIC TASTE; FOODS, DRUGS; SWEETENERS; POTASSIUM CHLORIDE BIORESEARCH, INC. (US) 1997-07-01 US disclosed
US-5631294-A PHENOXY- OR PHENYL-ALKANOIC ACIDS BIORESEARCH, INC. (US) 1997-05-20 US disclosed
US-5631038-A COMPOUNDS (TASTANDS) TO REDUCE OR ELIMINATE A BITTER OR METALLIC TASTE ARE ADDED TO FOODS CONTAINING SODIUM CHLORIDE BIORESEARCH, INC. (US) 1997-05-20 US disclosed
US-5631240-A KETONE BIORESEARCH, INC. (US) 1997-05-20 US disclosed
US-5631295-A 2-(4-METHOXYPHENOXY)PROPIONIC ACID, TAURINE, ASPARTYLPHENYL ALANINE, ASPARTYLTYROSINE AND DIHYDROXYBENZOIC ACID BIORESEARCH, INC. (US) 1997-05-20 US disclosed
US-5631299-A TAURINE OR AN ACCEPTABLE SALT (A TASTAND) TO REDUCE OR ELIMINATE A BITTER OR METALLIC TASTE; FOODS; DRUGS; SWEETENERS; POTASSIUM CHLORIDE BIORESEARCH, INC. (US) 1997-05-20 US disclosed
US-5631252-A Specific eatable taste modifiers BIORESEARCH, INC. (US) 1997-05-20 US disclosed
US-5631272-A SUBSTITUTED TRYPTAMINES BIORESEARCH, INC. (US) 1997-05-20 US disclosed
EP-0661932-A4 SPECIFIC EATABLE TASTE MODIFIERS. BIORESEARCH INC (US) 1996-06-05 EP disclosed
EP-0661932-A1 SPECIFIC EATABLE TASTE MODIFIERS BIORESEARCH, INC. (US) 1995-07-12 EP disclosed
WO-1993010677-A1 SPECIFIC EATABLE TASTE MODIFIERS BIORESEARCH, INC. (US) 1993-06-10 WO disclosed