SCHEMBL8215433

SCHEMBL8215433

Nc1cc(CS(=O)(=O)c2ccc(F)cc2)nc(-c2ccc(NC(=O)Nc3ccc(C(F)(F)F)cc3)cc2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 2/20 0.49
PIK3CA P42336 1/20 0.49
CA2 P00918 6/20 0.47
CA9 Q16790 6/20 0.47
CA12 O43570 5/20 0.47
CA1 P00915 5/20 0.47
MAPT P10636 2/20 0.47
MEN1 O00255 2/20 0.44
LMNA P02545 2/20 0.44
KMT2A Q03164 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CA4 P22748 1/20 0.42
CA7 P43166 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
ADORA1 P30542 1/20 0.42
EPHX2 P34913 3/20 0.41
AR P10275 1/20 0.41
KDR P35968 1/20 0.41
KDM1A O60341 1/20 0.40
RORC P51449 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8218182 0.87 PIK3CA (0.51) MTORPIK3CACA2CA9CA12
SCHEMBL8218786 0.86 PIK3CA (0.53) MTORPIK3CACA2CA9CA12
SCHEMBL8219760 0.86 PIK3CA (0.51) MTORPIK3CACA2CA9CA12
SCHEMBL8211599 0.85 PIK3CA (0.49) MTORPIK3CACA2CA9CA12
SCHEMBL8221081 0.84 PIK3CA (0.47) MTORPIK3CACA2CA9CA12
SCHEMBL8211601 0.84 PIK3CA (0.48) MTORPIK3CACA2CA9CA12
SCHEMBL8218892 0.84 PIK3CA (0.48) MTORPIK3CACA2CA9CA12
SCHEMBL8215437 0.84 PIK3CA (0.46) MTORPIK3CACA2CA9CA12
SCHEMBL8217566 0.83 PIK3CA (0.47) MTORPIK3CACA2CA9CA12
SCHEMBL11925678 0.83 PIK3CA (0.45) MTORPIK3CACA2CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008023159-A1 MORPHOLINO PYRIMIDINE DERIVATIVES USEFUL IN THE TREATMENT OF PROLIFERATIVE DISORDERS ASTRAZENECA AB (SE) 2008-02-28 WO disclosed