SCHEMBL8215510

SCHEMBL8215510

COC(=O)C(Cc1cc2c(cc1Cl)OCO2)CN(C)C

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
TAS1R3 Q7RTX0 5/20 0.38
TAS1R1 Q7RTX1 5/20 0.38
EDNRA P25101 1/20 0.38
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
UTS2R Q9UKP6 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6171617 0.85 SLC22A12 (0.38) BRS3CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6169213 0.84 BRS3 (0.40) BRS3CYP1A2CYP3A4CYP2D6CYP2C9
Iodide SCHEMBL8214551 0.82 BRS3 (0.40) BRS3CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6943904 0.73 CYP3A4 (0.44) BRS3CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6940934 0.71 CYP3A4 (0.42) BRS3CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL10871043 0.70 CYP3A4 (0.46) BRS3CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6584800 0.70 TAS1R3 (0.40) CYP3A4TAS1R3TAS1R1EDNRAMEN1
SCHEMBL13679360 0.70 KMT2A (0.45) MEN1KMT2AUTS2R
SCHEMBL8214818 0.69 HRH4 (0.42) BRS3CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL14707576 0.69 BRS3 (0.46) BRS3CYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6136842-A INHIBITION OF ENDOTHELIN-CONVERTING ENZYME HOECHST MARION ROUSSEL (FR) 2000-10-24 US disclosed