SCHEMBL6169213

SCHEMBL6169213

COC(=O)C(Cc1cc2c(cc1Cl)OCO2)C[N+](C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 1/20 0.40
CYP3A4 P08684 3/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
TAS1R3 Q7RTX0 5/20 0.37
TAS1R1 Q7RTX1 5/20 0.37
EDNRA P25101 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
NPC1 O15118 1/20 0.34
HTT P42858 1/20 0.34
RAB9A P51151 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL8214551 0.99 BRS3 (0.40) BRS3CYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL8215510 0.84 BRS3 (0.41) BRS3CYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL6943904 0.72 CYP3A4 (0.44) BRS3CYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL6171617 0.71 SLC22A12 (0.38) BRS3CYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL7373918 0.70 KMT2A (0.39) CYP3A4CYP1A2CYP2C9CYP2C19MEN1
SCHEMBL6940934 0.70 CYP3A4 (0.42) BRS3CYP3A4CYP1A2CYP2D6CYP2C9
Iodide SCHEMBL10568190 0.69 KMT2A (0.38) CYP3A4CYP1A2CYP2C9CYP2C19MEN1
SCHEMBL10871043 0.69 CYP3A4 (0.46) BRS3CYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL12404328 0.69 CRHBP (0.43) BRS3CYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL6584800 0.69 TAS1R3 (0.40) CYP3A4TAS1R3TAS1R1EDNRAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888341-B1 NOVEL SULPHUR DERIVATIVES COMPRISING AN AMIDE BOND, METHOD FOR PREPARING SAME, USE THEREOF AS DRUGS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH DERIVATIVES AVENTIS PHARMA SA (FR) 2005-11-30 EP disclosed
EP-0888341-A1 NOVEL SULPHUR DERIVATIVES COMPRISING AN AMIDE BOND, METHOD FOR PREPARING SAME, USE THEREOF AS DRUGS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH DERIVATIVES HOECHST MARION ROUSSEL (FR) 1999-01-07 EP disclosed
WO-1997032874-A1 NOVEL SULPHUR DERIVATIVES COMPRISING AN AMIDE BOND, METHOD FOR PREPARING SAME, USE THEREOF AS DRUGS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH DERIVATIVES HOECHST MARION ROUSSEL (FR) 1997-09-12 WO disclosed