SCHEMBL8215775

SCHEMBL8215775

[Pb].c1ccc2c(c1)CCCN2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.48
TSHR P16473 1/20 0.46
KDM4E B2RXH2 3/20 0.46
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
ALOX15 P16050 2/20 0.43
HSD17B10 Q99714 2/20 0.43
GAA P10253 2/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
THRB P10828 1/20 0.42
CASP1 P29466 1/20 0.42
HTT P42858 1/20 0.42
CASP7 P55210 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
NPC1 O15118 1/20 0.42
MAPK13 O15264 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29370549 0.98 MAPT (0.50) MAPTTSHRKDM4ECA12CA1
SCHEMBL27392334 0.98 MAPT (0.50) MAPTTSHRKDM4ECA12CA1
SCHEMBL18172 0.98 MAPT (0.50) MAPTTSHRKDM4ECA12CA1
SCHEMBL7259924 0.95 MAPT (0.48) MAPTTSHRKDM4ECA12CA1
Phosphine SCHEMBL241499 0.95 MAPT (0.48) MAPTTSHRKDM4ECA12CA1
SCHEMBL517747 0.95 MAPT (0.48) MAPTTSHRKDM4ECA12CA1
Methane SCHEMBL11211553 0.95 MAPT (0.48) MAPTTSHRKDM4ECA12CA1
Benzene SCHEMBL29053622 0.95 MAPT (0.50) MAPTTSHRKDM4ECA12CA1
Hydrochloric Acid SCHEMBL30018404 0.95 MAPT (0.48) MAPTTSHRKDM4ECA12CA1
Hydrochloric Acid SCHEMBL5370795 0.95 MAPT (0.48) MAPTTSHRKDM4ECA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1019720-A1 COMBINATORIAL PROCESS FOR PREPARING TETRAHYDROQUINOLINE LIBRARIES ELI LILLY AND COMPANY (US) 2000-07-19 EP disclosed
WO-1998027427-A1 COMBINATORIAL PROCESS FOR PREPARING TETRAHYDROQUINOLINE LIBRARIES ELI LILLY AND COMPANY (US) 1998-06-25 WO disclosed