SCHEMBL8217059

SCHEMBL8217059

ICc1cccn1Cc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.49
HDAC6 Q9UBN7 2/20 0.49
ALDH1A1 P00352 3/20 0.48
KDM4E B2RXH2 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
ADRA1D P25100 1/20 0.42
TNF P01375 1/20 0.42
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
DBH P09172 1/20 0.42
POLB P06746 2/20 0.41
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41
BRD4 O60885 2/20 0.41
BRD2 P25440 1/20 0.41
BRD3 Q15059 1/20 0.41
BRDT Q58F21 1/20 0.41
ALOX5 P09917 1/20 0.40
MAPT P10636 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27944822 0.82 ALDH1A1 (0.50) HDAC8HDAC6ALDH1A1KDM4EL3MBTL1
SCHEMBL27700003 0.82 ALDH1A1 (0.50) HDAC8HDAC6ALDH1A1KDM4EL3MBTL1
SCHEMBL28191937 0.80 HDAC8 (0.49) HDAC8HDAC6ALDH1A1KDM4EL3MBTL1
SCHEMBL1244069 0.80 HDAC8 (0.53) HDAC8HDAC6ALDH1A1KDM4EL3MBTL1
SCHEMBL3195611 0.80 HDAC8 (0.49) HDAC8HDAC6ALDH1A1KDM4EL3MBTL1
Iodomethane SCHEMBL7678454 0.77 ALDH1A1 (0.47) HDAC8HDAC6ALDH1A1KDM4EL3MBTL1
SCHEMBL7675436 0.76 ALDH1A1 (0.50) HDAC8HDAC6ALDH1A1KDM4EL3MBTL1
SCHEMBL12951910 0.76 AKR1B1 (0.50) HDAC8HDAC6ALDH1A1KDM4EL3MBTL1
SCHEMBL7674447 0.76 HDAC8 (0.45) HDAC8HDAC6ALDH1A1KDM4EL3MBTL1
SCHEMBL9767009 0.74 SIGMAR1 (0.52) HDAC8HDAC6ALDH1A1KDM4EL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008005456-A2 FUSED HETEROCYCLIC INHIBITORS OF D-AMINO ACID OXIDASE SEPRACOR INC. (US) 2008-01-10 WO disclosed