SCHEMBL8217835

SCHEMBL8217835

CC(C)(C)OC(=O)N1CCC2(CC1)C(=O)N(c1ccc(-c3ccccc3)cc1)C2c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 7/20 0.55
USP30 Q70CQ3 2/20 0.51
NR1H2 P55055 3/20 0.46
RXRA P19793 2/20 0.46
NR1H3 Q13133 2/20 0.46
GPR119 Q8TDV5 1/20 0.46
USP2 O75604 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
HSD17B10 Q99714 1/20 0.44
BACE1 P56817 2/20 0.43
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
ATM Q13315 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8212694 0.93 TRPV1 (0.61) TRPV1USP30GPR119ALOX15TSHR
SCHEMBL8217839 0.93 CACNA1H (0.49) TRPV1USP30
SCHEMBL8226841 0.91 TRPV1 (0.54) TRPV1USP30GPR119
SCHEMBL8224724 0.91 HDAC1 (0.53) TRPV1USP30NR1H2RXRANR1H3
SCHEMBL8227841 0.87 TRPV1 (0.55) TRPV1USP30GPR119ALOX15TSHR
SCHEMBL14263432 0.86 CACNA1H (0.54) TRPV1GPR119
SCHEMBL8225731 0.86 CACNA1H (0.48) TRPV1USP30GPR119
SCHEMBL8207926 0.85 TRPV1 (0.51) TRPV1USP30GPR119ALOX15TSHR
SCHEMBL8228184 0.85 CACNA1H (0.53) TRPV1USP30
SCHEMBL8218928 0.84 HDAC1 (0.56) TRPV1USP30GPR119ALDH1A1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080076750-A1 Azetidinone Derivatives and Methods of Use Thereof SCHERING CORPORATION 2008-03-27 US disclosed
US-20080076750-A1 Azetidinone Derivatives and Methods of Use Thereof SCHERING CORPORATION 2008-03-27 US disclosed
WO-2008033460-A2 TREATING PAIN, DIABETES, AND LIPID METABOLISM DISORDERS SCHERING CORPORATION (US) 2008-03-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080076750-A1 Azetidinone Derivatives and Methods of Use Thereof LIPC, CES1, ZDHHC20 TRPV1 438/4885USP30 1448/4885NR1H2 36/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.