SCHEMBL8218149

SCHEMBL8218149

NCCCNc1nc(=O)c2ccccc2[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 2/20 0.47
TRPC3 Q13507 1/20 0.47
TRPC4 Q9UBN4 1/20 0.47
TRPC5 Q9UL62 1/20 0.47
TSHR P16473 1/20 0.42
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
PRKD3 O94806 4/20 0.40
PRKCG P05129 4/20 0.40
PRKCB P05771 4/20 0.40
PRKCA P17252 4/20 0.40
PRKCH P24723 4/20 0.40
PRKCI P41743 4/20 0.40
PRKCE Q02156 4/20 0.40
PRKCQ Q04759 4/20 0.40
PRKCZ Q05513 4/20 0.40
PRKCD Q05655 4/20 0.40
PRKD1 Q15139 4/20 0.40
PIM1 P11309 1/20 0.40
APP P05067 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6034415 0.79 BCHE (0.72) BCHETRPC3TRPC4TRPC5TSHR
SCHEMBL7217251 0.79 ALDH1A1 (0.48) TSHRKDM4EALDH1A1APPHSD17B10
SCHEMBL18934416 0.77 KDM4E (0.70) BCHETRPC3TRPC4TRPC5KDM4E
SCHEMBL6856197 0.77 ALDH1A1 (0.44) TSHRKDM4EALDH1A1APPHSD17B10
SCHEMBL30013315 0.77 ALDH1A1 (0.44) TSHRKDM4EALDH1A1APPHSD17B10
SCHEMBL178850 0.76 MARS1 (0.46)
SCHEMBL178859 0.76 MARS1 (0.51) KCNH2
SCHEMBL4640893 0.75 BCHE (0.70) BCHETRPC3TRPC4TRPC5TSHR
SCHEMBL6439777 0.74 BCHE (0.68) BCHETRPC3TRPC4TRPC5TSHR
SCHEMBL5668076 0.72 MARS1 (0.59)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000071524-A1 2-NH-PYRIDONES AND PYRIMIDONES AS MRS INHIBITORS SMITHKLINE BEECHAM PLC (GB) 2000-11-30 WO disclosed