SCHEMBL8218501

SCHEMBL8218501

N#CN(CS(=O)(=O)c1ccc(N)cc1)C(N)=Nc1ccncc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLG P00747 1/20 0.36
NOS3 P29474 2/20 0.35
NOS1 P29475 2/20 0.35
NOS2 P35228 2/20 0.35
GAA P10253 2/20 0.34
F2 P00734 2/20 0.33
PRSS1 P07477 2/20 0.33
PRSS2 P07478 2/20 0.33
PRSS3 P35030 2/20 0.33
LMNA P02545 2/20 0.33
AGO2 Q9UKV8 1/20 0.33
TSHR P16473 2/20 0.30
NAMPT P43490 1/20 0.30
KDM4E B2RXH2 1/20 0.30
POLB P06746 1/20 0.30
MAPT P10636 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
ALDH1A1 P00352 1/20 0.30
NT5E P21589 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8218500 0.88 CYP17A1 (0.36) PLGNOS3NOS1NOS2NAMPT
SCHEMBL8200238 0.79 PLG (0.40) PLGNOS3NOS1NOS2GAA
SCHEMBL504667 0.72 PLG (0.44) PLGNOS3NOS1NOS2
SCHEMBL504588 0.72 PLG (0.44) PLGNOS3NOS1NOS2
SCHEMBL9299302 0.70 PLG (0.42) PLGNOS3NOS1NOS2KDM4E
SCHEMBL504564 0.69 PLG (0.41) PLGNOS3NOS1NOS2F2
SCHEMBL8200233 0.68 CYP17A1 (0.45) PLGNOS3NOS1NOS2ALDH1A1
SCHEMBL2351953 0.60 KMT2A (0.71) GAALMNATSHRTDP1L3MBTL1
SCHEMBL5745307 0.60 GAA (0.55) GAAF2PRSS1PRSS2PRSS3
SCHEMBL7082360 0.59 CYP3A4 (0.47) GAALMNAAGO2TSHRNAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000061561-A1 CYANOGUANIDINE COMPOUNDS SHIONOGI BIORESEARCH CORP. (US) 2000-10-19 WO disclosed