SCHEMBL8219623

SCHEMBL8219623

Nc1nc(-c2ccccn2)cc2cc[c]cc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 3/20 0.42
CCR5 P51681 3/20 0.42
CCR8 P51685 3/20 0.42
KDM4E B2RXH2 7/20 0.42
ALDH1A1 P00352 3/20 0.42
HPGD P15428 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
GLA P06280 2/20 0.42
GAA P10253 2/20 0.42
POLB P06746 2/20 0.42
HCRTR1 O43613 1/20 0.42
MEN1 O00255 1/20 0.42
MAPT P10636 1/20 0.42
TSHR P16473 1/20 0.42
KMT2A Q03164 1/20 0.42
ADORA3 P0DMS8 7/20 0.42
LMNA P02545 3/20 0.41
HSP90AA1 P07900 2/20 0.41
METAP1 P53582 2/20 0.41
CYP1A2 P05177 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8221653 0.88 CCR1 (0.42) CCR1CCR5CCR8KDM4EALDH1A1
SCHEMBL8222632 0.88 ADORA2A (0.35) KDM4EALDH1A1HPGDSMN1; SMN2GLA
SCHEMBL10389484 0.81 ADORA3 (0.55) CCR1CCR5CCR8KDM4EALDH1A1
SCHEMBL11371057 0.79 KDM4E (0.49) CCR1CCR5CCR8KDM4EALDH1A1
SCHEMBL6090464 0.76 SYK (0.36) KDM4EALDH1A1HPGDSMN1; SMN2GLA
SCHEMBL8219421 0.74 KDM4E (0.47) KDM4EALDH1A1HPGDSMN1; SMN2GLA
SCHEMBL11381433 0.73 SYK (0.58) CCR1CCR5CCR8KDM4EALDH1A1
SCHEMBL11367963 0.73 CCR1 (0.45) CCR1CCR5CCR8KDM4EALDH1A1
SCHEMBL11367019 0.72 ADORA3 (0.50) CCR1CCR5CCR8KDM4EALDH1A1
SCHEMBL11361335 0.72 ADORA3 (0.50) CCR1CCR5CCR8KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188120-B2 Lactam-containing compounds and derivatives thereof as factor Xa inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2012-05-29 US disclosed