SCHEMBL8220948

SCHEMBL8220948

O=C1CCC2(CC1)C(=O)Nc1cc(Cl)ccc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNKS O95271 1/20 0.51
TNKS2 Q9H2K2 1/20 0.51
PGR P06401 4/20 0.48
PDE7A Q13946 1/20 0.47
PKM P14618 1/20 0.44
CMA1 P23946 1/20 0.44
AHR P35869 1/20 0.44
TP53 P04637 1/20 0.41
MDM2 Q00987 1/20 0.41
IP6K1 Q92551 6/20 0.41
AKR1B1 P15121 1/20 0.40
IP6K3 Q96PC2 1/20 0.40
IP6K2 Q9UHH9 1/20 0.40
OTUD7B Q6GQQ9 1/20 0.39
GHSR Q92847 1/20 0.39
HTR1A P08908 1/20 0.39
HTR2A P28223 1/20 0.39
HTR7 P34969 1/20 0.39
HTR6 P50406 1/20 0.39
SRD5A1 P18405 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26666490 0.90 PGR (0.56) TNKSTNKS2PGRPDE7APKM
SCHEMBL30701457 0.87 PGR (0.58) TNKSTNKS2PGRPDE7APKM
SCHEMBL30701438 0.87 PGR (0.58) TNKSTNKS2PGRPDE7APKM
SCHEMBL11641780 0.87 PGR (0.58) TNKSTNKS2PGRPDE7APKM
SCHEMBL4715820 0.85 PGR (0.59) TNKSTNKS2PGRPDE7APKM
SCHEMBL20955697 0.84 PKM (0.53) TNKSTNKS2PGRPDE7APKM
SCHEMBL23778352 0.82 CYP3A4 (0.43) AKR1B1
SCHEMBL12437085 0.82 TNKS (0.45) TNKSTNKS2PGRPDE7APKM
SCHEMBL30898646 0.81 CMA1 (0.44) TNKSTNKS2PGRCMA1AHR
SCHEMBL23778308 0.81 TNKS (0.50) TNKSTNKS2PGRHTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008055812-A1 SPIROINDOLINONE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-05-15 WO disclosed