Chlorotrianisene

Chlorotrianisene

SCHEMBL8225

COc1ccc(C(Cl)=C(c2ccc(OC)cc2)c2ccc(OC)cc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ESR2

The experimentally established mechanism targets of Chlorotrianisene. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 1.00
ALDH1A1 P00352 2/20 1.00
SMN1; SMN2 Q16637 2/20 1.00
KDM4E B2RXH2 1/20 1.00
LMNA P02545 1/20 1.00
ESR1 P03372 1/20 1.00
ADORA3 P0DMS8 1/20 1.00
MAPT P10636 1/20 1.00
TSHR P16473 1/20 1.00
MAPK1 P28482 1/20 1.00
CYP2C19 P33261 1/20 1.00
ADRA1A P35348 1/20 1.00
HIF1A Q16665 1/20 1.00
NPSR1 Q6W5P4 1/20 1.00
HSD17B10 Q99714 1/20 1.00
TCF4 P15884 1/20 0.58
CTNNB1 P35222 1/20 0.58
CA1 P00915 5/20 0.56
CA2 P00918 5/20 0.56
CES2 O00748 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Chlorotrianisene SCHEMBL7349593 1.00 HPGD (1.00) HPGDALDH1A1SMN1; SMN2KDM4ELMNA
SCHEMBL8613998 0.92 ESR1 (0.85) HPGDALDH1A1SMN1; SMN2KDM4ELMNA
SCHEMBL23358693 0.92 ESR1 (0.85) HPGDALDH1A1SMN1; SMN2KDM4ELMNA
SCHEMBL23358692 0.92 ESR1 (0.85) HPGDALDH1A1SMN1; SMN2KDM4ELMNA
Chlorotrianisene SCHEMBL4928327 0.90 MAPT (0.81) HPGDALDH1A1SMN1; SMN2KDM4ELMNA
SCHEMBL12710298 0.87 SMN1; SMN2 (0.76) HPGDALDH1A1SMN1; SMN2KDM4ELMNA
Chlorotrianisene SCHEMBL28258939 0.86 ALDH1A1 (0.73) HPGDALDH1A1SMN1; SMN2KDM4ELMNA
SCHEMBL22773016 0.84 TSHR (0.72) HPGDALDH1A1SMN1; SMN2KDM4ELMNA
Chlorotrianisene SCHEMBL5528225 0.83 MAPT (0.69) HPGDALDH1A1SMN1; SMN2KDM4ELMNA
SCHEMBL2957320 0.83 ALDH1A1 (0.70) HPGDALDH1A1SMN1; SMN2KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 25176 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4735116-A2 ANTI-TRAILR2 ANTIGEN-BINDING PROTEINS AND USES THEREOF ODYSSEY THERAPEUTICS, INC. (US) 2026-05-06 EP claimed
EP-4711364-A1 FUSED PYRROLE RING OR FUSED PYRIDINE RING COMPOUND Pharmaengine, Inc. (TW) 2026-03-18 EP claimed
EP-4701737-A2 MTA-COOPERATIVE PRMT5 INHIBITOR Pharmaengine, Inc. (TW) 2026-03-04 EP claimed
EP-4695235-A1 NOVEL GSPT1 DEGRADER AND USE THEREOF Cyrus Therapeutics Inc. (KR) 2026-02-18 EP claimed
WO-2025227007-A1 METHODS AND COMPOSITIONS FOR INHIBITION OF DIHYDROOROTATE DEHYDROGENASE OHIO STATE INNOVATION FOUNDATION (US) 2025-10-30 WO claimed
US-12454519-B2 Substituted N-(2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-5-yl)arylsulfonamide analogs as modulators of cereblon protein ST. JUDE CHILDREN'S RESEARCH HOSPITAL, INC. (US) 2025-10-28 US claimed
US-12454518-B2 Substituted N-(2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-5-yl)arylsulfonamide analogs as modulators of cereblon protein ST. JUDE CHILDREN'S RESEARCH HOSPITAL, INC. (US) 2025-10-28 US claimed
EP-3710001-B1 COMPOUNDS AND METHODS FOR REGULATING, LIMITING, OR INHIBITING AVIL EXPRESSION UNIV VIRGINIA PATENT FOUNDATION (US) 2025-06-18 EP claimed
EP-3324856-B1 SHEAR-THINNING COMPOSITIONS AS AN INTRAVASCULAR EMBOLIC AGENT BRIGHAM & WOMENS HOSPITAL INC (US) 2025-04-23 EP claimed
WO-2025080751-A2 ANTI-CDH17 ANTIGEN-BINDING PROTEINS AND USES THEREOF ODYSSEY THERAPEUTICS, INC. (US) 2025-04-17 WO claimed
WO-1991005603-A1 DEVICE FOR IMPROVING THE EVAPORATION AND/OR THE HOMOGENIZING OF A MIXTURE OF A GASEUS AND/OR LIQUID FLUID HERAIL RENE (FR) 1991-05-02 WO claimed
US-4729999-A MENOPAUSE, SIDE EFFECT PREVENTION BCM TECHNOLOGIES (US) 1988-03-08 US claimed
US-4712765-A Apparatus for producing coated panels STELLA WERKE AG (CH) 1987-12-15 US claimed
EP-0247394-A2 Sealed thrust ball bearing KOYO SEIKO CO., LTD. (JP) 1987-12-02 EP claimed
EP-0234988-A1 Propulsion unit combustion chamber and its assembly method SOCIETE EUROPEENNE DE PROPULSION (FR) 1987-09-02 EP claimed
EP-0178043-A1 Power supply for electroluminescent panels LUMINESCENT ELECTRONICS, INC. (US) 1986-04-16 EP claimed
EP-0108584-A1 Syringes Dentsply Limited (GB) 1984-05-16 EP claimed
WO-1984001607-A1 MOTION TRANSMITTING DEVICES QUADRANT DRIVE (NL) 1984-04-26 WO claimed
US-4310523-A Combined antiestrogens and antigonadotropically effective antiandrogens for the prophylaxis and therapy of hyperplasia of the prostate SCHERING AKTIENGESELLSCHAFT (DE) 1982-01-12 US claimed
EP-0010964-A1 Ravidomycin, process of preparation and pharmaceutical compositions containing same AYERST, MCKENNA AND HARRISON INC. (CA) 1980-05-14 EP claimed