SCHEMBL8225217

SCHEMBL8225217

O=C(c1ccc2oc(NCc3cccc(Cl)c3)nc2c1)N(CCCn1ccnc1)Cc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
THRB P10828 5/20 0.52
NAMPT P43490 7/20 0.45
HDAC1 Q13547 1/20 0.43
KCNA5 P22460 1/20 0.43
CYP3A4 P08684 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8220847 0.95 THRB (0.54) THRBNAMPTHDAC1CYP3A4HDAC6
SCHEMBL8228578 0.94 THRB (0.50) THRBNAMPTHDAC1KCNA5CYP3A4
SCHEMBL8226119 0.92 THRB (0.51) THRBNAMPTHDAC1KCNA5CYP3A4
SCHEMBL8226260 0.90 THRB (0.50) THRBNAMPTHDAC1KCNA5CYP3A4
SCHEMBL8229319 0.87 THRB (0.55) THRBHDAC1HDAC6NPC1
SCHEMBL8229336 0.85 THRB (0.55) THRBNAMPTHDAC1HDAC6NPC1
SCHEMBL8226265 0.84 THRB (0.56) THRBHDAC1HDAC6NPC1
SCHEMBL8231029 0.84 THRB (0.54) THRBHDAC1HDAC6NPC1
SCHEMBL8219815 0.83 THRB (0.61) THRBHDAC1HDAC6NPC1
SCHEMBL8226029 0.83 THRB (0.53) THRBHDAC1HDAC6NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007140982-A1 SUBSTITUTED BENZOXAZOLES BAYER HEALTHCARE AG (DE) 2007-12-13 WO disclosed