SCHEMBL8230253

SCHEMBL8230253

C=CSc1ccncc1N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC1 P19801 2/20 0.44
AOC3 Q16853 2/20 0.44
IMPDH2 P12268 3/20 0.43
GAA P10253 2/20 0.38
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
MEN1 O00255 1/20 0.37
KDM6B O15054 1/20 0.37
KDM4A O75164 1/20 0.37
MAPT P10636 1/20 0.37
THRB P10828 1/20 0.37
KMT2A Q03164 1/20 0.37
KDM4D Q6B0I6 1/20 0.37
KDM4C Q9H3R0 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CA12 O43570 6/20 0.35
CA1 P00915 6/20 0.35
CA2 P00918 6/20 0.35
CA9 Q16790 6/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8223054 0.77 AOC1 (0.41) AOC1AOC3IMPDH2GAAKDM4E
SCHEMBL16326502 0.76 CA12 (0.33) IMPDH2TDP1CA12CA1CA2
SCHEMBL19225669 0.76 IMPDH2 (0.36) IMPDH2CA12CA1CA2CA9
SCHEMBL20777739 0.74
SCHEMBL16702153 0.73 HASPIN (0.43) AOC1AOC3IMPDH2GAAKDM4E
SCHEMBL11023159 0.72
SCHEMBL31354791 0.72
SCHEMBL19225663 0.72 IMPDH2 (0.36) IMPDH2
SCHEMBL4169429 0.72 AOC3 (0.44) AOC1AOC3GAAKDM4EALDH1A1
SCHEMBL16712907 0.72 AOC1 (0.44) AOC1AOC3IMPDH2GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007144128-A1 PYRROLIDINE COMPOUNDS AS RENIN INHIBITORS NOVARTIS AG (CH) 2007-12-21 WO disclosed